calcium channel, voltage-dependent, N type, alpha 1B subunit |
GUANETHIDINE |
Calcium Channel Type L, Benzothiazepine |
54% |
NoneNone |
NoneNone |
View
|
calcium channel, voltage-dependent, alpha2/delta subunit 1 |
GUANETHIDINE |
Calcium Channel Type L, Benzothiazepine |
54% |
NoneNone |
NoneNone |
View
|
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 |
PERGOLIDE |
Serotonin Transporter |
54% |
NoneNone |
NoneNone |
View
|
Cytochrom P450-2C19 monooxygenase |
FLUCONAZOLE |
CYP450-2C19 Inhibition |
54% |
NoneNone |
NoneNone |
View
|
adenosine A2a receptor |
GW-1929 |
Adenosine A2A |
54% |
37.254uM |
20.915uM |
View
|
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) |
KETOCONAZOLE |
CYP450-2C9 Inhibition |
54% |
NoneNone |
NoneNone |
View
|
cytochrome P450, family 2, subfamily C, polypeptide 9 |
KETOCONAZOLE |
CYP450-2C9 Inhibition |
54% |
NoneNone |
NoneNone |
View
|
mitogen activated protein kinase 1 |
TYRPHOSTIN A23 |
Protein Serine/Threonine Kinase, ERK2 |
54% |
NoneNone |
NoneNone |
View
|
mitogen-activated protein kinase 1 |
TYRPHOSTIN A23 |
Protein Serine/Threonine Kinase, ERK2 |
54% |
NoneNone |
NoneNone |
View
|
mitogen activated protein kinase 3 |
AURANOFIN |
Protein Serine/Threonine Kinase, ERK1 |
54% |
NoneNone |
NoneNone |
View
|
mitogen-activated protein kinase 3 |
AURANOFIN |
Protein Serine/Threonine Kinase, ERK1 |
54% |
NoneNone |
NoneNone |
View
|
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 4 |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
gamma-aminobutyric acid A receptor, gamma 1 |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
gamma-aminobutyric acid A receptor, pi |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
AT hook, DNA binding motif, containing 1 (DBSS) |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
gamma-aminobutyric acid A receptor, theta |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
gamma-aminobutyric acid A receptor, gamma 2 |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
sodium channel associated protein 1 |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel associated protein 2 |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type III, beta |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type I, alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type IX, alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type VII, alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
amiloride-sensitive cation channel 5, intestinal |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type III, beta |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type VIII, alpha polypeptide |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type XI, alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type I, beta |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type 10, alpha polypeptide |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type IV, alpha polypeptide |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type V, alpha polypeptide |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type II, beta |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, nonvoltage-gated 1 alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, nonvoltage-gated 1 gamma |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, nonvoltage-gated 1 beta |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type 2, alpha 1 polypeptide |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type XI, alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, nonvoltage-gated 1, gamma |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, nonvoltage-gated 1, delta |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, nonvoltage-gated 1 alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type X, alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type IX, alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage gated, type VIII, alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type VII, alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type IV, beta |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type IV, alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type III, alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type II, beta |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type II, alpha 2 |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type I, beta |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type I, alpha |
CLOZAPINE |
Sodium Channel, Site 2 |
53% |
NoneNone |
NoneNone |
View
|
mitogen activated protein kinase 3 |
THIOGUANINE |
Protein Serine/Threonine Kinase, ERK1 |
53% |
5.516uM |
NoneNone |
View
|
mitogen-activated protein kinase 3 |
THIOGUANINE |
Protein Serine/Threonine Kinase, ERK1 |
53% |
5.516uM |
NoneNone |
View
|
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 |
DEXTROMETHORPHAN |
Adrenergic, Norepinephrine Transporter |
53% |
NoneNone |
NoneNone |
View
|
adrenergic receptor, alpha 1a |
DEXTROMETHORPHAN |
Adrenergic alpha1A |
53% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type II, beta |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, nonvoltage-gated 1 alpha |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, nonvoltage-gated 1 gamma |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, nonvoltage-gated 1 beta |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, voltage-gated, type 2, alpha 1 polypeptide |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, voltage-gated, type XI, alpha |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, nonvoltage-gated 1, gamma |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, nonvoltage-gated 1, delta |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, nonvoltage-gated 1 alpha |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, voltage-gated, type X, alpha |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, voltage-gated, type IX, alpha |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, voltage gated, type VIII, alpha |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, voltage-gated, type VII, alpha |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) |
DICLOFENAC |
Sodium Channel, Site 2 |
53% |
53.142uM |
47.644uM |
View
|
phosphodiesterase 3B |
MICONAZOLE |
Phosphodiesterase PDE3 |
53% |
73.911uM |
NoneNone |
View
|
sodium channel, voltage-gated, type 2, alpha 1 polypeptide |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type XI, alpha |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, nonvoltage-gated 1, gamma |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, nonvoltage-gated 1, delta |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, nonvoltage-gated 1 alpha |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type X, alpha |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type IX, alpha |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage gated, type VIII, alpha |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type VII, alpha |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type IV, beta |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type IV, alpha |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type III, alpha |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type II, beta |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type II, alpha 2 |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type I, beta |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type I, alpha |
S-(-)-PROPRANOLOL |
Sodium Channel, Site 2 |
52% |
NoneNone |
NoneNone |
View
|
5-hydroxytryptamine (serotonin) receptor 2B |
DISULFIRAM |
Serotonin 5-HT2B |
52% |
34.547uM |
21.984uM |
View
|
adrenergic receptor, alpha 1a |
KETOCONAZOLE |
Adrenergic alpha1A |
52% |
35.729uM |
14.462uM |
View
|
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 |
SIMVASTATIN |
Dopamine Transporter |
52% |
NoneNone |
NoneNone |
View
|
Cytochrom P450-1A2 monooxygenase |
AURANOFIN |
CYP450-1A2 Inhibition |
52% |
NoneNone |
NoneNone |
View
|
matrix metallopeptidase 9 |
CAMPTOTHECIN |
Protease, Matrix Metalloprotease-9 (MMP-9) |
52% |
NoneNone |
NoneNone |
View
|
matrix metalloproteinase 9 (gelatinase B, 92kDa gelatinase, 92kDa type IV collagenase) |
CAMPTOTHECIN |
Protease, Matrix Metalloprotease-9 (MMP-9) |
52% |
NoneNone |
NoneNone |
View
|
mitogen activated protein kinase 14 |
DIETHYLSTILBESTROL |
Protein Serine/Threonine Kinase, p38alpha |
52% |
32.903uM |
NoneNone |
View
|
mitogen-activated protein kinase 14 |
DIETHYLSTILBESTROL |
Protein Serine/Threonine Kinase, p38alpha |
52% |
32.903uM |
NoneNone |
View
|
estrogen receptor 1 |
4-OCTYLPHENOL |
Estrogen ERalpha |
52% |
27.674uM |
7.907uM |
View
|
estrogen receptor 1 |
4-OCTYLPHENOL |
Estrogen ERalpha |
52% |
27.674uM |
7.907uM |
View
|
5-hydroxytryptamine (serotonin) receptor 1A |
BACITRACIN |
Serotonin 5-HT1A |
52% |
NoneNone |
NoneNone |
View
|
dopamine receptor D4 |
ALPHA-ERGOCRYPTINE |
Dopamine D4.2 |
52% |
NoneNone |
NoneNone |
View
|
dopamine receptor D3 |
CLOSANTEL |
Dopamine D3 |
52% |
NoneNone |
NoneNone |
View
|
mitogen activated protein kinase 14 |
GRAMICIDIN |
Protein Serine/Threonine Kinase, p38alpha |
52% |
NoneNone |
NoneNone |
View
|
mitogen-activated protein kinase 14 |
GRAMICIDIN |
Protein Serine/Threonine Kinase, p38alpha |
52% |
NoneNone |
NoneNone |
View
|
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 |
MAPROTILINE |
Serotonin Transporter |
52% |
NoneNone |
NoneNone |
View
|
adrenergic receptor, alpha 1b |
BUSPIRONE |
Adrenergic alpha1B |
52% |
NoneNone |
NoneNone |
View
|
adrenergic receptor, alpha 2a |
BUSPIRONE |
Adrenergic alpha2A |
52% |
NoneNone |
NoneNone |
View
|
chemokine (C-C motif) receptor 5 |
OXCARBAZEPINE |
Chemokine CCR5 |
52% |
NoneNone |
NoneNone |
View
|
Cytochrom P450-1A2 monooxygenase |
ERGOTAMINE |
CYP450-1A2 Inhibition |
52% |
NoneNone |
NoneNone |
View
|
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 4 |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
gamma-aminobutyric acid A receptor, gamma 1 |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
gamma-aminobutyric acid A receptor, pi |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
AT hook, DNA binding motif, containing 1 (DBSS) |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
gamma-aminobutyric acid A receptor, theta |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
gamma-aminobutyric acid A receptor, gamma 2 |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 6 |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 5 |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
gamma-aminobutyric acid A receptor, alpha 2 |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
gamma-aminobutyric acid A receptor, alpha 1 |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 2 |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 1 |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
gamma-aminobutyric acid A receptor, delta |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 3 |
VX-745 |
GABAA, Benzodiazepine, Central |
52% |
11.986uM |
9.767uM |
View
|
dopamine receptor D1A |
TERCONAZOLE |
Dopamine D1 |
52% |
25.48uM |
12.74uM |
View
|
androgen receptor |
NELFINAVIR |
Testosterone |
52% |
36.389uM |
24.259uM |
View
|
5-hydroxytryptamine (serotonin) receptor 1B |
TERCONAZOLE |
Serotonin 5-HT1B |
52% |
89.897uM |
40.862uM |
View
|
sodium channel, voltage-gated, type II, alpha 2 |
ERGOTAMINE |
Sodium Channel, Site 2 |
51% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type I, beta |
ERGOTAMINE |
Sodium Channel, Site 2 |
51% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type I, alpha |
ERGOTAMINE |
Sodium Channel, Site 2 |
51% |
NoneNone |
NoneNone |
View
|
sodium channel, voltage-gated, type V, alpha polypeptide |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type II, beta |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, nonvoltage-gated 1 alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, nonvoltage-gated 1 gamma |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, nonvoltage-gated 1 beta |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type 2, alpha 1 polypeptide |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type XI, alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, nonvoltage-gated 1, gamma |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, nonvoltage-gated 1, delta |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, nonvoltage-gated 1 alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type X, alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type IX, alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage gated, type VIII, alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type VII, alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type IV, beta |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type IV, alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type III, alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type II, beta |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type II, alpha 2 |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type I, beta |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type I, alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type IV, beta |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel associated protein 1 |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel associated protein 2 |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type III, beta |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type I, alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type IX, alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type VII, alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
amiloride-sensitive cation channel 5, intestinal |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type III, beta |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type VIII, alpha polypeptide |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type XI, alpha |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type I, beta |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type 10, alpha polypeptide |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
sodium channel, voltage-gated, type IV, alpha polypeptide |
VX-745 |
Sodium Channel, Site 2 |
51% |
26.533uM |
23.788uM |
View
|
adrenergic receptor, alpha 2a |
HYDROXYPROGESTERONE |
Adrenergic alpha2A |
51% |
NoneNone |
NoneNone |
View
|
melanocortin 5 receptor |
PIPAMAZINE |
Melanocortin MC5 |
51% |
NoneNone |
NoneNone |
View
|
dopamine receptor D3 |
FENOFIBRATE |
Dopamine D3 |
51% |
137.533uM |
46.709uM |
View
|
Cytochrom P450-2C19 monooxygenase |
DANAZOL |
CYP450-2C19 Inhibition |
51% |
NoneNone |
NoneNone |
View
|
matrix metalloproteinase 1 (interstitial collagenase) |
CAMPTOTHECIN |
Protease, Matrix Metalloprotease-1 (MMP-1) |
51% |
NoneNone |
NoneNone |
View
|
progesterone receptor |
BETA-ESTRADIOL |
Progesterone |
51% |
32.559uM |
4.247uM |
View
|
progesterone receptor |
BETA-ESTRADIOL |
Progesterone |
51% |
32.559uM |
4.247uM |
View
|
adenosine A1 receptor |
NOCODAZOLE |
Adenosine A1 |
51% |
50.33uM |
29.433uM |
View
|
thromboxane A synthase 1 |
LIPOPOLYSACCHARIDE E. COLI O55:B5 |
Thromboxane Synthetase |
51% |
NoneNone |
NoneNone |
View
|
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) |
LIPOPOLYSACCHARIDE E. COLI O55:B5 |
Thromboxane Synthetase |
51% |
NoneNone |
NoneNone |
View
|
glutamate receptor, ionotropic, N-methyl D-aspartate 2D |
AMANTADINE |
Glutamate, NMDA, Phencyclidine |
51% |
31.983uM |
21.666uM |
View
|
glutamate receptor, ionotropic, NMDA2C |
AMANTADINE |
Glutamate, NMDA, Phencyclidine |
51% |
31.983uM |
21.666uM |
View
|
glutamate receptor, ionotropic, N-methyl D-aspartate 2B |
AMANTADINE |
Glutamate, NMDA, Phencyclidine |
51% |
31.983uM |
21.666uM |
View
|
glutamate receptor, ionotropic, N-methyl D-aspartate 2A |
AMANTADINE |
Glutamate, NMDA, Phencyclidine |
51% |
31.983uM |
21.666uM |
View
|
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 6 |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 5 |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
gamma-aminobutyric acid A receptor, alpha 2 |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
gamma-aminobutyric acid A receptor, alpha 1 |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 2 |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 1 |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
gamma-aminobutyric acid A receptor, delta |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 3 |
LY-294002 |
GABAA, Benzodiazepine, Central |
54% |
21.411uM |
17.446uM |
View
|
calcium channel, voltage-dependent, gamma subunit 4 |
MIFEPRISTONE |
Calcium Channel Type L, Phenylalkylamine |
54% |
16.01uM |
15.559uM |
View
|
calcium channel, voltage-dependent, gamma subunit 3 |
MIFEPRISTONE |
Calcium Channel Type L, Phenylalkylamine |
54% |
16.01uM |
15.559uM |
View
|
calcium channel, voltage-dependent, gamma subunit 2 |
MIFEPRISTONE |
Calcium Channel Type L, Phenylalkylamine |
54% |
16.01uM |
15.559uM |
View
|
calcium channel, voltage-dependent, gamma subunit 1 |
MIFEPRISTONE |
Calcium Channel Type L, Phenylalkylamine |
54% |
16.01uM |
15.559uM |
View
|
calcium channel, voltage-dependent, beta 4 subunit |
MIFEPRISTONE |
Calcium Channel Type L, Phenylalkylamine |
54% |
16.01uM |
15.559uM |
View
|
calcium channel, voltage-dependent, beta 3 subunit |
MIFEPRISTONE |
Calcium Channel Type L, Phenylalkylamine |
54% |
16.01uM |
15.559uM |
View
|
calcium channel, voltage-dependent, beta 2 subunit |
MIFEPRISTONE |
Calcium Channel Type L, Phenylalkylamine |
54% |
16.01uM |
15.559uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1S subunit |
MIFEPRISTONE |
Calcium Channel Type L, Phenylalkylamine |
54% |
16.01uM |
15.559uM |
View
|
calcium channel, voltage-dependent, alpha 1F subunit |
MIFEPRISTONE |
Calcium Channel Type L, Phenylalkylamine |
54% |
16.01uM |
15.559uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1D subunit |
MIFEPRISTONE |
Calcium Channel Type L, Phenylalkylamine |
54% |
16.01uM |
15.559uM |
View
|