Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
potassium voltage-gated channel, subfamily H (eag-related), member 6 PENTAMIDINE Potassium Channel HERG 54% 15.7215uM 12.8802uM View
potassium voltage-gated channel, subfamily H (eag-related), member 7 PENTAMIDINE Potassium Channel HERG 54% 15.7215uM 12.8802uM View
potassium voltage-gated channel, subfamily H (eag-related), member 2 PENTAMIDINE Potassium Channel HERG 54% 15.7215uM 12.8802uM View
potassium voltage-gated channel, subfamily H (eag-related), member 5 PENTAMIDINE Potassium Channel HERG 54% 15.7215uM 12.8802uM View
potassium voltage-gated channel, subfamily H (eag-related), member 3 PENTAMIDINE Potassium Channel HERG 54% 15.7215uM 12.8802uM View
potassium voltage-gated channel, subfamily H (eag-related), member 4 PENTAMIDINE Potassium Channel HERG 54% 15.7215uM 12.8802uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 PENTAMIDINE Potassium Channel HERG 54% 15.7215uM 12.8802uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 PENTAMIDINE Potassium Channel HERG 54% 15.7215uM 12.8802uM View
cytochrome P450, family 3, subfamily a, polypeptide 13 FLUORESCEIN CYP450-3A4 Inhibition 54% NoneNone NoneNone View
chemokine (C-C motif) receptor 2 TRANS-PLATINUM(II)DIAMMINE DICHLORIDE Chemokine CCR2B 54% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 3,3',5-TRIIODO-L-THYRONINE Adrenergic, Norepinephrine Transporter 54% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase FLUNARIZINE CYP450-2C19 Inhibition 54% NoneNone NoneNone View
adrenergic receptor, alpha 1a SULOCTIDIL Adrenergic alpha1A 54% NoneNone NoneNone View
Sigma-2 Receptor AMBROXOL Sigma2 54% NoneNone NoneNone View
Protein-tyrosine kinase, Fyn FLUNARIZINE Protein Tyrosine Kinase, Fyn 54% NoneNone NoneNone View
dopamine receptor D4 DOMPERIDONE Dopamine D4.2 54% NoneNone NoneNone View
dopamine receptor D3 4-NONYLPHENOL Dopamine D3 54% NoneNone NoneNone View
dopamine receptor D3 HYDROXYPROGESTERONE Dopamine D3 54% NoneNone NoneNone View
dopamine receptor D1A HYDROXYPROGESTERONE Dopamine D1 54% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase MOCLOBEMIDE CYP450-2D6 Inhibition 54% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase SELEGILINE CYP450-2D6 Inhibition 54% NoneNone NoneNone View
Cytochrom P450-2D6 monooxygenase MOSAPRIDE CYP450-2D6 Inhibition 54% NoneNone NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) ANISINDIONE CYP450-2C9 Inhibition 54% NoneNone NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 ANISINDIONE CYP450-2C9 Inhibition 54% NoneNone NoneNone View
acetylcholinesterase (YT blood group) HYDROXYPROGESTERONE Acetylcholinesterase 54% NoneNone NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase HYDROXYPROGESTERONE Acetylcholinesterase 54% NoneNone NoneNone View
acetylcholinesterase HYDROXYPROGESTERONE Acetylcholinesterase 54% NoneNone NoneNone View
ATPase, Na+/K+ transporting, beta 3 polypeptide 3,3',4',5-TETRACHLOROSALICYLANILIDE ATPase, Na+/K+ 54% NoneNone NoneNone View
ATPase, Na+/K+ transporting, beta 2 polypeptide 3,3',4',5-TETRACHLOROSALICYLANILIDE ATPase, Na+/K+ 54% NoneNone NoneNone View
ATPase, (Na+)/K+ transporting, beta 4 polypeptide 3,3',4',5-TETRACHLOROSALICYLANILIDE ATPase, Na+/K+ 54% NoneNone NoneNone View
ATPase, Na+/K+ transporting, alpha 4 polypeptide 3,3',4',5-TETRACHLOROSALICYLANILIDE ATPase, Na+/K+ 54% NoneNone NoneNone View
ATPase, Na+/K+ transporting, alpha 3 polypeptide 3,3',4',5-TETRACHLOROSALICYLANILIDE ATPase, Na+/K+ 54% NoneNone NoneNone View
ATPase, Na+/K+ transporting, alpha 2 polypeptide 3,3',4',5-TETRACHLOROSALICYLANILIDE ATPase, Na+/K+ 54% NoneNone NoneNone View
ATPase, Na+/K+ transporting, alpha 1 polypeptide 3,3',4',5-TETRACHLOROSALICYLANILIDE ATPase, Na+/K+ 54% NoneNone NoneNone View
ATPase, Na+/K+ transporting, beta 1 polypeptide 3,3',4',5-TETRACHLOROSALICYLANILIDE ATPase, Na+/K+ 54% NoneNone NoneNone View
adrenergic receptor, alpha 2a BUFLOMEDIL Imidazoline I2, Central 54% NoneNone NoneNone View
adrenergic receptor, alpha 2c (Non-specific probe) BUFLOMEDIL Imidazoline I2, Central 54% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 AMITRAZ Dopamine Transporter 54% NoneNone NoneNone View
5-hydroxytryptamine (serotonin) receptor 1B AMITRAZ Serotonin 5-HT1B 54% NoneNone NoneNone View
estrogen receptor 1 ETHISTERONE Estrogen ERalpha 54% NoneNone NoneNone View
estrogen receptor 1 ETHISTERONE Estrogen ERalpha 54% NoneNone NoneNone View
adrenergic receptor, alpha 1a DIPHENIDOL Adrenergic alpha1A 54% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 PROCHLORPERAZINE Calcium Channel Type L, Benzothiazepine 53% NoneNone NoneNone View
leukotriene B4 receptor 2 PIOGLITAZONE Leukotriene B4 53% 86.922uM 22.055uM View
leukotriene B4 receptor PIOGLITAZONE Leukotriene B4 53% 86.922uM 22.055uM View
leukotriene B4 receptor PIOGLITAZONE Leukotriene B4 53% 86.922uM 22.055uM View
leukotriene B4 receptor 2 PIOGLITAZONE Leukotriene B4 53% 86.922uM 22.055uM View
prostaglandin-endoperoxide synthase 2 PIROXICAM Cyclooxygenase COX-2 53% NoneNone NoneNone View
prostaglandin-endoperoxide synthase 2 (prostaglandin G/H synthase and cyclooxygenase) PIROXICAM Cyclooxygenase COX-2 53% NoneNone NoneNone View
melanocortin 4 receptor VINORELBINE Melanocortin MC4 52.5% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 alpha PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type X, alpha PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type IX, alpha PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage gated, type VIII, alpha PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type VII, alpha PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, beta PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, alpha PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type III, alpha PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type II, beta PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type II, alpha 2 PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type I, beta PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type I, alpha PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, beta PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel associated protein 1 PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel associated protein 2 PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type III, beta PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
sodium channel, voltage-gated, type I, alpha PRIMAQUINE Sodium Channel, Site 2 52% NoneNone NoneNone View
Sigma-2 Receptor PROMETHAZINE Sigma2 52% NoneNone NoneNone View
Cytochrom P450-1A2 monooxygenase TRIOXSALEN CYP450-1A2 Inhibition 52% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 RESVERATROL Dopamine Transporter 52% NoneNone NoneNone View
prostaglandin-endoperoxide synthase 1 VALDECOXIB Cyclooxygenase COX-1 52% NoneNone NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) VALDECOXIB Cyclooxygenase COX-1 52% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase BAY 11-7085 CYP450-2C19 Inhibition 52% NoneNone NoneNone View
Cytochrom P450-1A2 monooxygenase DROPERIDOL CYP450-1A2 Inhibition 52% NoneNone NoneNone View
melanocortin 4 receptor EMETINE Melanocortin MC4 52% NoneNone NoneNone View
dopamine receptor 2 DISULFIRAM Dopamine D2L 52% 23.018uM 7.673uM View
5-hydroxytryptamine (serotonin) receptor 2C ALOSETRON Serotonin 5-HT2C 52% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 S-(-)-PROPRANOLOL Calcium Channel Type L, Phenylalkylamine 52% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 S-(-)-PROPRANOLOL Calcium Channel Type L, Phenylalkylamine 52% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 S-(-)-PROPRANOLOL Calcium Channel Type L, Phenylalkylamine 52% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 S-(-)-PROPRANOLOL Calcium Channel Type L, Phenylalkylamine 52% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 S-(-)-PROPRANOLOL Calcium Channel Type L, Phenylalkylamine 52% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 7 LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 LACIDIPINE Calcium Channel Type L, Phenylalkylamine 51% NoneNone NoneNone View
ATPase, Na+/K+ transporting, beta 1 polypeptide TRIBROMSALAN ATPase, Na+/K+ 51% NoneNone NoneNone View
ATPase, Na+/K+ transporting, beta 3 polypeptide TRIBROMSALAN ATPase, Na+/K+ 51% NoneNone NoneNone View
ATPase, Na+/K+ transporting, beta 2 polypeptide TRIBROMSALAN ATPase, Na+/K+ 51% NoneNone NoneNone View
ATPase, (Na+)/K+ transporting, beta 4 polypeptide TRIBROMSALAN ATPase, Na+/K+ 51% NoneNone NoneNone View
ATPase, Na+/K+ transporting, alpha 4 polypeptide TRIBROMSALAN ATPase, Na+/K+ 51% NoneNone NoneNone View
ATPase, Na+/K+ transporting, alpha 3 polypeptide TRIBROMSALAN ATPase, Na+/K+ 51% NoneNone NoneNone View
ATPase, Na+/K+ transporting, alpha 2 polypeptide TRIBROMSALAN ATPase, Na+/K+ 51% NoneNone NoneNone View
ATPase, Na+/K+ transporting, alpha 1 polypeptide TRIBROMSALAN ATPase, Na+/K+ 51% NoneNone NoneNone View
tachykinin receptor 2 CANDESARTAN Tachykinin NK2 51% NoneNone NoneNone View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) SB-203580 Protein Tyrosine Kinase, HER2 Receptor 51% 18.896uM NoneNone View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) SB-203580 Protein Tyrosine Kinase, HER2 Receptor 51% 18.896uM NoneNone View
androgen receptor CLOMIPHENE Testosterone 51% NoneNone NoneNone View
opioid receptor, kappa 1 DOXAZOSIN Opiate kappa 51% NoneNone NoneNone View
Sigma-2 Receptor DISULFIRAM Sigma2 51% 75.564uM 46.501uM View
Sigma-2 Receptor MOSAPRIDE Sigma2 51% NoneNone NoneNone View
lymphocyte protein tyrosine kinase (mapped) BROMOCRIPTINE Protein Tyrosine Kinase, Lck 51% NoneNone NoneNone View
adrenergic receptor, alpha 2a CITALOPRAM Adrenergic alpha2A 51% NoneNone NoneNone View
adrenergic receptor, beta 1 LYSERGOL Adrenergic beta1 51% NoneNone NoneNone View
adrenergic, beta-1-, receptor LYSERGOL Adrenergic beta1 51% NoneNone NoneNone View
adrenergic receptor, alpha 1d (Non-specific probe) METHYSERGIDE Adrenergic alpha1D 51% NoneNone NoneNone View
cholinergic receptor, muscarinic 1 LORATADINE Muscarinic M1 51% NoneNone NoneNone View
5-hydroxytryptamine receptor 6 4-(PHENYLMETHYL)-1-[2-(TRIFLUOROMETHYL)BENZOYL]-PIPERIDINE Serotonin 5-HT6 51% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase MC 258717 CYP450-2C19 Inhibition 51% NoneNone NoneNone View
A3 adenosine receptor RWJ-68354 Adenosine A3 51% NoneNone NoneNone View
adrenergic receptor, alpha 1a RWJ-68354 Adrenergic alpha1A 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 7 MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit MITOTANE Calcium Channel Type L, Dihydropyridine 51% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 gamma ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 beta ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type XI, alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, gamma ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, delta ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type X, alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type IX, alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage gated, type VIII, alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type VII, alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, beta ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type III, alpha ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
sodium channel, voltage-gated, type II, beta ERGOTAMINE Sodium Channel, Site 2 51% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit MOSAPRIDE Calcium Channel Type L, Phenylalkylamine 50% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit MOSAPRIDE Calcium Channel Type L, Phenylalkylamine 50% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit MOSAPRIDE Calcium Channel Type L, Phenylalkylamine 50% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 MOSAPRIDE Calcium Channel Type L, Phenylalkylamine 50% NoneNone NoneNone View
histamine receptor H 2 BROMOCRIPTINE Histamine H2 50% NoneNone NoneNone View
thromboxane A synthase 1 BROMOCRIPTINE Thromboxane Synthetase 50% NoneNone NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) BROMOCRIPTINE Thromboxane Synthetase 50% NoneNone NoneNone View
adenosine A2a receptor MITOTANE Adenosine A2A 50% NoneNone NoneNone View
epidermal growth factor receptor ITRACONAZOLE Protein Tyrosine Kinase, EGF Receptor 50% NoneNone NoneNone View
matrix metallopeptidase 9 GADOPENTETATE DIMEGLUMINE Protease, Matrix Metalloprotease-9 (MMP-9) 50% NoneNone NoneNone View
matrix metalloproteinase 9 (gelatinase B, 92kDa gelatinase, 92kDa type IV collagenase) GADOPENTETATE DIMEGLUMINE Protease, Matrix Metalloprotease-9 (MMP-9) 50% NoneNone NoneNone View
5-hydroxytryptamine receptor 6 PHENTOLAMINE Serotonin 5-HT6 50% NoneNone NoneNone View
caspase 1 SULFASALAZINE Protease, Caspase 1 50% 28.812uM NoneNone View
caspase 1, apoptosis-related cysteine protease (interleukin 1, beta, convertase) SULFASALAZINE Protease, Caspase 1 50% 28.812uM NoneNone View
caspase 3, apoptosis related cysteine protease SULFASALAZINE Protease, Caspase 1 50% 28.812uM NoneNone View
caspase 2 SULFASALAZINE Protease, Caspase 1 50% 28.812uM NoneNone View
caspase 7 SULFASALAZINE Protease, Caspase 1 50% 28.812uM NoneNone View
caspase 6 SULFASALAZINE Protease, Caspase 1 50% 28.812uM NoneNone View
Cytochrom P450-2D6 monooxygenase DROPERIDOL CYP450-2D6 Inhibition 50% NoneNone NoneNone View
mitogen activated protein kinase 14 ANTIMYCIN A Protein Serine/Threonine Kinase, p38alpha 50% NoneNone NoneNone View
mitogen-activated protein kinase 14 ANTIMYCIN A Protein Serine/Threonine Kinase, p38alpha 50% NoneNone NoneNone View
phosphodiesterase 4A, cAMP specific TROGLITAZONE Phosphodiesterase PDE4 50% NoneNone NoneNone View
phosphodiesterase 4C, cAMP-specific TROGLITAZONE Phosphodiesterase PDE4 50% NoneNone NoneNone View
phosphodiesterase 4D TROGLITAZONE Phosphodiesterase PDE4 50% NoneNone NoneNone View
phosphodiesterase 4B, cAMP specific TROGLITAZONE Phosphodiesterase PDE4 50% NoneNone NoneNone View
arachidonate 15-lipoxygenase CAFFEIC ACID PHENETHYL ESTER Lipoxygenase 15-LO 50% NoneNone NoneNone View
arachidonate 15-lipoxygenase CAFFEIC ACID PHENETHYL ESTER Lipoxygenase 15-LO 50% NoneNone NoneNone View
sodium channel, voltage-gated, type VIII, alpha polypeptide FLAVOXATE Sodium Channel, Site 2 50% NoneNone NoneNone View
sodium channel, voltage-gated, type XI, alpha FLAVOXATE Sodium Channel, Site 2 50% NoneNone NoneNone View
sodium channel, voltage-gated, type I, beta FLAVOXATE Sodium Channel, Site 2 50% NoneNone NoneNone View
sodium channel, voltage-gated, type 10, alpha polypeptide FLAVOXATE Sodium Channel, Site 2 50% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, alpha polypeptide FLAVOXATE Sodium Channel, Site 2 50% NoneNone NoneNone View
sodium channel, voltage-gated, type V, alpha polypeptide FLAVOXATE Sodium Channel, Site 2 50% NoneNone NoneNone View