Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
glutamate receptor, ionotropic, N-methyl D-aspartate 2A CLOTRIMAZOLE Glutamate, NMDA, Agonism 88% 13.064uM 11.82uM View
N-methyl-D-aspartate receptor 1 (Grin1) gene, exons 1 through 6 and partial cds; alternatively spliced (Rn.) CLOTRIMAZOLE Glutamate, NMDA, Agonism 88% 13.064uM 11.82uM View
glutamate receptor, ionotropic, N-methyl-D-aspartate 3B CLOTRIMAZOLE Glutamate, NMDA, Agonism 88% 13.064uM 11.82uM View
5-hydroxytryptamine (serotonin) receptor 2C CLOTRIMAZOLE Serotonin 5-HT2C 88% 14.472uM 7.581uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 AMIODARONE Adrenergic, Norepinephrine Transporter 88% 2.271uM 2.252uM View
thromboxane A synthase 1 TAMOXIFEN Thromboxane Synthetase 88% .916uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) TAMOXIFEN Thromboxane Synthetase 88% .916uM NoneNone View
A3 adenosine receptor TAMOXIFEN Adenosine A3 88% 3.701uM 2.092uM View
calcium channel, voltage-dependent, gamma subunit 8 DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, gamma subunit 7 DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, gamma subunit 6 DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, gamma subunit 5 DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, gamma subunit 4 DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, gamma subunit 3 DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, gamma subunit 2 DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, gamma subunit 1 DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, beta 4 subunit DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, beta 3 subunit DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, beta 2 subunit DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, gamma subunit 5 CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, gamma subunit 4 CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, gamma subunit 3 CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, gamma subunit 2 CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, gamma subunit 1 CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, beta 4 subunit CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, beta 3 subunit CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, beta 2 subunit CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, alpha 1F subunit CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, beta 1 subunit CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 CINNARIZINE Calcium Channel Type L, Benzothiazepine 87% .823uM .732uM View
cytochrome P450, family 3, subfamily a, polypeptide 13 PHENYLHYDRAZINE CYP450-3A4 Inhibition 87% .9uM NoneNone View
Cytochrom P450-2D6 monooxygenase PROPRANOLOL CYP450-2D6 Inhibition 87% 2uM NoneNone View
Cytochrom P450-2D6 monooxygenase LANSOPRAZOLE CYP450-2D6 Inhibition 87% 5.3148uM NoneNone View
arachidonate 15-lipoxygenase, second type VINBLASTINE Lipoxygenase 15-LO 87% 5.037uM NoneNone View
arachidonate 15-lipoxygenase VINBLASTINE Lipoxygenase 15-LO 87% 5.037uM NoneNone View
arachidonate 15-lipoxygenase VINBLASTINE Lipoxygenase 15-LO 87% 5.037uM NoneNone View
adrenergic receptor, beta 2 DOBUTAMINE Adrenergic beta2 87% 1.517uM 1.043uM View
adrenergic receptor, alpha 2a METHYLERGONOVINE Adrenergic alpha2A 87% 1.59uM .596uM View
adrenergic receptor, alpha 1d (Non-specific probe) CLONIDINE Adrenergic alpha1D 87% 1.21uM .595uM View
adrenergic receptor, alpha 1d (Non-specific probe) BUSPIRONE Adrenergic alpha1D 87% 1.077uM .529uM View
dopamine receptor D1A ERGOTAMINE Dopamine D1 87% 1.728uM .864uM View
histamine receptor H 1 PROMAZINE Histamine H1, Central 87% .003435uM .000399uM View
thromboxane A synthase 1 NELFINAVIR Thromboxane Synthetase 87% 21.11uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) NELFINAVIR Thromboxane Synthetase 87% 21.11uM NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, gamma subunit 4 NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, gamma subunit 3 NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, gamma subunit 2 NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, gamma subunit 1 NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, beta 4 subunit NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, beta 3 subunit NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, beta 2 subunit NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, alpha 1F subunit NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, beta 1 subunit NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
cholinergic receptor, muscarinic 1 CLOMIPHENE Muscarinic M1 86% 1.628uM .392uM View
calcium channel, voltage-dependent, gamma subunit 8 CLOMIPHENE Calcium Channel Type L, Phenylalkylamine 86% .754uM .733uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit TIRILAZAD Calcium Channel Type L, Phenylalkylamine 86% 2.496uM 2.427uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit TIRILAZAD Calcium Channel Type L, Phenylalkylamine 86% 2.496uM 2.427uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit TIRILAZAD Calcium Channel Type L, Phenylalkylamine 86% 2.496uM 2.427uM View
calcium channel, voltage-dependent, beta 1 subunit TIRILAZAD Calcium Channel Type L, Phenylalkylamine 86% 2.496uM 2.427uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit TIRILAZAD Calcium Channel Type L, Phenylalkylamine 86% 2.496uM 2.427uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit TIRILAZAD Calcium Channel Type L, Phenylalkylamine 86% 2.496uM 2.427uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 TIRILAZAD Calcium Channel Type L, Phenylalkylamine 86% 2.496uM 2.427uM View
opioid receptor, delta 1 PACLITAXEL Opiate delta 86% 4.202uM 1.481uM View
opioid receptor, sigma 1 AMITRIPTYLINE Sigma1 86% 1.031uM .433uM View
adrenergic receptor, alpha 2a AMOXAPINE Adrenergic alpha2A 86% 1.314uM .493uM View
calcium channel, voltage-dependent, gamma subunit 8 U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, gamma subunit 7 U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, gamma subunit 6 U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, gamma subunit 5 U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, gamma subunit 4 U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, gamma subunit 3 U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, gamma subunit 2 U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, gamma subunit 1 U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, beta 4 subunit U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, beta 3 subunit U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, beta 2 subunit U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, alpha 1F subunit U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
5-hydroxytryptamine (serotonin) receptor 1A BW-723C86 Serotonin 5-HT1A 86% 1.1278uM .6445uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 BUPROPION Dopamine Transporter 86% 1.0338uM .8214uM View
tachykinin receptor 2 4-NONYLPHENOL Tachykinin NK2 86% 4.514uM 1.505uM View
sodium channel, voltage-gated, type IV, beta THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel associated protein 1 THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel associated protein 2 THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type III, beta THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type I, alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type IX, alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type VII, alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
amiloride-sensitive cation channel 5, intestinal THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type III, beta THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type XI, alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type I, beta THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type 10, alpha polypeptide THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type IV, alpha polypeptide THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type V, alpha polypeptide THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type II, beta THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, nonvoltage-gated 1 alpha THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, nonvoltage-gated 1 gamma THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, nonvoltage-gated 1 beta THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide THIORIDAZINE Sodium Channel, Site 2 86% 2.056uM 1.876uM View
calcium channel, voltage-dependent, beta 4 subunit FLUPHENAZINE Calcium Channel Type L, Phenylalkylamine 89% 2.534uM 2.464uM View
calcium channel, voltage-dependent, beta 3 subunit FLUPHENAZINE Calcium Channel Type L, Phenylalkylamine 89% 2.534uM 2.464uM View
calcium channel, voltage-dependent, beta 2 subunit FLUPHENAZINE Calcium Channel Type L, Phenylalkylamine 89% 2.534uM 2.464uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit FLUPHENAZINE Calcium Channel Type L, Phenylalkylamine 89% 2.534uM 2.464uM View
calcium channel, voltage-dependent, alpha 1F subunit FLUPHENAZINE Calcium Channel Type L, Phenylalkylamine 89% 2.534uM 2.464uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit FLUPHENAZINE Calcium Channel Type L, Phenylalkylamine 89% 2.534uM 2.464uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit FLUPHENAZINE Calcium Channel Type L, Phenylalkylamine 89% 2.534uM 2.464uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit FLUPHENAZINE Calcium Channel Type L, Phenylalkylamine 89% 2.534uM 2.464uM View
calcium channel, voltage-dependent, beta 1 subunit FLUPHENAZINE Calcium Channel Type L, Phenylalkylamine 89% 2.534uM 2.464uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit FLUPHENAZINE Calcium Channel Type L, Phenylalkylamine 89% 2.534uM 2.464uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit FLUPHENAZINE Calcium Channel Type L, Phenylalkylamine 89% 2.534uM 2.464uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 FLUPHENAZINE Calcium Channel Type L, Phenylalkylamine 89% 2.534uM 2.464uM View
adrenergic receptor, alpha 2a DOXEPIN Adrenergic alpha2A 89% 1.335uM .501uM View
histamine receptor H 2 HALOPERIDOL Histamine H2 89% 1.166uM 1.147uM View
adrenergic receptor, alpha 2b MONTELUKAST Adrenergic alpha2C 89% 5.279uM .767uM View
adrenergic receptor, alpha 2c (Non-specific probe) MONTELUKAST Adrenergic alpha2C 89% 5.279uM .767uM View
5-hydroxytryptamine (serotonin) receptor 2B CITALOPRAM Serotonin 5-HT2B 89% 1.839uM 1.171uM View
cholinergic receptor, muscarinic 3 MIANSERIN Muscarinic M3 89% 1.405uM .298uM View
cholinergic receptor, muscarinic 1 MIANSERIN Muscarinic M1 89% 1.423uM .343uM View
mitogen activated protein kinase 14 MC 258717 Protein Serine/Threonine Kinase, p38alpha 89% 2.272uM NoneNone View
mitogen-activated protein kinase 14 MC 258717 Protein Serine/Threonine Kinase, p38alpha 89% 2.272uM NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) 1-(2-METHOXYBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE CYP450-2C9 Inhibition 89% 2uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 1-(2-METHOXYBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE CYP450-2C9 Inhibition 89% 2uM NoneNone View
adrenergic receptor, alpha 2a 1-NAPHTHYL ISOTHIOCYANATE Adrenergic alpha2A 89% 6.272uM 2.352uM View
cholinergic receptor, muscarinic 4 QUINACRINE Muscarinic M4 89% 1.983uM .277uM View
cholinergic receptor, muscarinic 4 KETOTIFEN Muscarinic M4 89% 1.009uM .141uM View
adrenergic receptor, alpha 2a SELEGILINE Adrenergic alpha2A 89% 1.798uM .674uM View
monoamine oxidase A NABUMETONE Monoamine Oxidase MAOA 89% .998uM NoneNone View
monoamine oxidase A NABUMETONE Monoamine Oxidase MAOA 89% .998uM NoneNone View
adrenergic receptor, alpha 2a NORTRIPTYLINE Adrenergic alpha2A 89% .732uM .275uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 OLANZAPINE Serotonin Transporter 89% 1.033uM .549uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 NORETHINDRONE Serotonin Transporter 89% 4.537uM 2.411uM View
5-hydroxytryptamine (serotonin) receptor 1A NORTRIPTYLINE Serotonin 5-HT1A 89% 1.868uM 1.068uM View
adrenergic receptor, alpha 2a OXYMETAZOLINE Imidazoline I2, Central 89% .027uM .018uM View
adrenergic receptor, alpha 2c (Non-specific probe) OXYMETAZOLINE Imidazoline I2, Central 89% .027uM .018uM View
dopamine receptor 2 EBASTINE Dopamine D2L 89% 1.1491uM .383uM View
A3 adenosine receptor EBASTINE Adenosine A3 89% 3.1953uM 1.8061uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 4 CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
gamma-aminobutyric acid A receptor, gamma 1 CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
gamma-aminobutyric acid A receptor, pi CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
AT hook, DNA binding motif, containing 1 (DBSS) CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
gamma-aminobutyric acid A receptor, theta CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
gamma-aminobutyric acid A receptor, gamma 2 CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 6 CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 5 CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
gamma-aminobutyric acid A receptor, alpha 2 CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
gamma-aminobutyric acid A receptor, alpha 1 CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 2 CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 1 CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
gamma-aminobutyric acid A receptor, delta CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, alpha 1F subunit DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, beta 1 subunit DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 DICYCLOMINE Calcium Channel Type L, Benzothiazepine 88% 1.736uM 1.543uM View
3-hydroxy-3-methylglutaryl-Coenzyme A reductase CISAPRIDE HMG-CoA Reductase 88% 3.37uM NoneNone View
3-hydroxy-3-methylglutaryl-Coenzyme A reductase CISAPRIDE HMG-CoA Reductase 88% 3.37uM NoneNone View
dopamine receptor 2 CISAPRIDE Dopamine D2L 88% .473uM .158uM View
dopamine receptor D1A CARVEDILOL Dopamine D1 88% 1.498uM .749uM View
adrenergic receptor, beta 3 TIMOLOL Adrenergic beta3 88% .452uM .339uM View
cholinergic receptor, muscarinic 5 FLUOXETINE Muscarinic M5 88% 1.358uM .976uM View
phosphodiesterase 3B CILOSTAZOL Phosphodiesterase PDE3 88% .271uM NoneNone View
phosphodiesterase 3A CILOSTAZOL Phosphodiesterase PDE3 88% .271uM NoneNone View
adrenergic receptor, alpha 2b TICLOPIDINE Adrenergic alpha2C 88% 1.175uM .171uM View
adrenergic receptor, alpha 2c (Non-specific probe) TICLOPIDINE Adrenergic alpha2C 88% 1.175uM .171uM View
A3 adenosine receptor SULINDAC SULFIDE Adenosine A3 88% 7.231uM 4.087uM View
prostaglandin-endoperoxide synthase 1 MONOBENZONE Cyclooxygenase COX-1 88% 1.019uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) MONOBENZONE Cyclooxygenase COX-1 88% 1.019uM NoneNone View
calcium channel, voltage-dependent, beta 4 subunit HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
sodium channel, voltage-gated, type IX, alpha BENZTROPINE Sodium Channel, Site 2 88% 1.68uM 1.533uM View
adrenergic receptor, beta 1 LISURIDE Adrenergic beta1 88% .559uM .323uM View
adrenergic, beta-1-, receptor LISURIDE Adrenergic beta1 88% .559uM .323uM View
adrenergic receptor, alpha 2b MAPROTILINE Adrenergic alpha2C 88% 3.044uM .442uM View
adrenergic receptor, alpha 2c (Non-specific probe) MAPROTILINE Adrenergic alpha2C 88% 3.044uM .442uM View
dopamine receptor D1A IVERMECTIN Dopamine D1 88% 4.5148uM 2.2574uM View
5-hydroxytryptamine (serotonin) receptor 2C PYRILAMINE Serotonin 5-HT2C 88% 1.13uM .592uM View
mitogen activated protein kinase 14 VX-745 Protein Serine/Threonine Kinase, p38alpha 88% .643uM NoneNone View
mitogen-activated protein kinase 14 VX-745 Protein Serine/Threonine Kinase, p38alpha 88% .643uM NoneNone View
adrenergic receptor, alpha 1b ROXITHROMYCIN Adrenergic alpha1B 88% .989uM .548uM View
adenosine A2a receptor SILDENAFIL Adenosine A2A 88% .253uM .142uM View