glutamate receptor, ionotropic, N-methyl D-aspartate 2A |
CLOTRIMAZOLE |
Glutamate, NMDA, Agonism |
88% |
13.064uM |
11.82uM |
View
|
N-methyl-D-aspartate receptor 1 (Grin1) gene, exons 1 through 6 and partial cds; alternatively spliced (Rn.) |
CLOTRIMAZOLE |
Glutamate, NMDA, Agonism |
88% |
13.064uM |
11.82uM |
View
|
glutamate receptor, ionotropic, N-methyl-D-aspartate 3B |
CLOTRIMAZOLE |
Glutamate, NMDA, Agonism |
88% |
13.064uM |
11.82uM |
View
|
5-hydroxytryptamine (serotonin) receptor 2C |
CLOTRIMAZOLE |
Serotonin 5-HT2C |
88% |
14.472uM |
7.581uM |
View
|
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 |
AMIODARONE |
Adrenergic, Norepinephrine Transporter |
88% |
2.271uM |
2.252uM |
View
|
thromboxane A synthase 1 |
TAMOXIFEN |
Thromboxane Synthetase |
88% |
.916uM |
NoneNone |
View
|
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) |
TAMOXIFEN |
Thromboxane Synthetase |
88% |
.916uM |
NoneNone |
View
|
A3 adenosine receptor |
TAMOXIFEN |
Adenosine A3 |
88% |
3.701uM |
2.092uM |
View
|
calcium channel, voltage-dependent, gamma subunit 8 |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, gamma subunit 7 |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, gamma subunit 6 |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, gamma subunit 5 |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, gamma subunit 4 |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, gamma subunit 3 |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, gamma subunit 2 |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, gamma subunit 1 |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, beta 4 subunit |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, beta 3 subunit |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, beta 2 subunit |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, gamma subunit 5 |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, gamma subunit 4 |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, gamma subunit 3 |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, gamma subunit 2 |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, gamma subunit 1 |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, beta 4 subunit |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, beta 3 subunit |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, beta 2 subunit |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1S subunit |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, alpha 1F subunit |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1D subunit |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1C subunit |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, beta 1 subunit |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1E subunit |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, N type, alpha 1B subunit |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
calcium channel, voltage-dependent, alpha2/delta subunit 1 |
CINNARIZINE |
Calcium Channel Type L, Benzothiazepine |
87% |
.823uM |
.732uM |
View
|
cytochrome P450, family 3, subfamily a, polypeptide 13 |
PHENYLHYDRAZINE |
CYP450-3A4 Inhibition |
87% |
.9uM |
NoneNone |
View
|
Cytochrom P450-2D6 monooxygenase |
PROPRANOLOL |
CYP450-2D6 Inhibition |
87% |
2uM |
NoneNone |
View
|
Cytochrom P450-2D6 monooxygenase |
LANSOPRAZOLE |
CYP450-2D6 Inhibition |
87% |
5.3148uM |
NoneNone |
View
|
arachidonate 15-lipoxygenase, second type |
VINBLASTINE |
Lipoxygenase 15-LO |
87% |
5.037uM |
NoneNone |
View
|
arachidonate 15-lipoxygenase |
VINBLASTINE |
Lipoxygenase 15-LO |
87% |
5.037uM |
NoneNone |
View
|
arachidonate 15-lipoxygenase |
VINBLASTINE |
Lipoxygenase 15-LO |
87% |
5.037uM |
NoneNone |
View
|
adrenergic receptor, beta 2 |
DOBUTAMINE |
Adrenergic beta2 |
87% |
1.517uM |
1.043uM |
View
|
adrenergic receptor, alpha 2a |
METHYLERGONOVINE |
Adrenergic alpha2A |
87% |
1.59uM |
.596uM |
View
|
adrenergic receptor, alpha 1d (Non-specific probe) |
CLONIDINE |
Adrenergic alpha1D |
87% |
1.21uM |
.595uM |
View
|
adrenergic receptor, alpha 1d (Non-specific probe) |
BUSPIRONE |
Adrenergic alpha1D |
87% |
1.077uM |
.529uM |
View
|
dopamine receptor D1A |
ERGOTAMINE |
Dopamine D1 |
87% |
1.728uM |
.864uM |
View
|
histamine receptor H 1 |
PROMAZINE |
Histamine H1, Central |
87% |
.003435uM |
.000399uM |
View
|
thromboxane A synthase 1 |
NELFINAVIR |
Thromboxane Synthetase |
87% |
21.11uM |
NoneNone |
View
|
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) |
NELFINAVIR |
Thromboxane Synthetase |
87% |
21.11uM |
NoneNone |
View
|
calcium channel, voltage-dependent, gamma subunit 5 |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, gamma subunit 4 |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, gamma subunit 3 |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, gamma subunit 2 |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, gamma subunit 1 |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, beta 4 subunit |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, beta 3 subunit |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, beta 2 subunit |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1S subunit |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, alpha 1F subunit |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1D subunit |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1C subunit |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, beta 1 subunit |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1E subunit |
NELFINAVIR |
Calcium Channel Type L, Dihydropyridine |
87% |
9.84uM |
6.324uM |
View
|
cholinergic receptor, muscarinic 1 |
CLOMIPHENE |
Muscarinic M1 |
86% |
1.628uM |
.392uM |
View
|
calcium channel, voltage-dependent, gamma subunit 8 |
CLOMIPHENE |
Calcium Channel Type L, Phenylalkylamine |
86% |
.754uM |
.733uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1D subunit |
TIRILAZAD |
Calcium Channel Type L, Phenylalkylamine |
86% |
2.496uM |
2.427uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1C subunit |
TIRILAZAD |
Calcium Channel Type L, Phenylalkylamine |
86% |
2.496uM |
2.427uM |
View
|
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
TIRILAZAD |
Calcium Channel Type L, Phenylalkylamine |
86% |
2.496uM |
2.427uM |
View
|
calcium channel, voltage-dependent, beta 1 subunit |
TIRILAZAD |
Calcium Channel Type L, Phenylalkylamine |
86% |
2.496uM |
2.427uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1E subunit |
TIRILAZAD |
Calcium Channel Type L, Phenylalkylamine |
86% |
2.496uM |
2.427uM |
View
|
calcium channel, voltage-dependent, N type, alpha 1B subunit |
TIRILAZAD |
Calcium Channel Type L, Phenylalkylamine |
86% |
2.496uM |
2.427uM |
View
|
calcium channel, voltage-dependent, alpha2/delta subunit 1 |
TIRILAZAD |
Calcium Channel Type L, Phenylalkylamine |
86% |
2.496uM |
2.427uM |
View
|
opioid receptor, delta 1 |
PACLITAXEL |
Opiate delta |
86% |
4.202uM |
1.481uM |
View
|
opioid receptor, sigma 1 |
AMITRIPTYLINE |
Sigma1 |
86% |
1.031uM |
.433uM |
View
|
adrenergic receptor, alpha 2a |
AMOXAPINE |
Adrenergic alpha2A |
86% |
1.314uM |
.493uM |
View
|
calcium channel, voltage-dependent, gamma subunit 8 |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, gamma subunit 7 |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, gamma subunit 6 |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, gamma subunit 5 |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, gamma subunit 4 |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, gamma subunit 3 |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, gamma subunit 2 |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, gamma subunit 1 |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, beta 4 subunit |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, beta 3 subunit |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, beta 2 subunit |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1S subunit |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, alpha 1F subunit |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1D subunit |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1C subunit |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
U-78517F |
Calcium Channel Type L, Dihydropyridine |
86% |
1.659uM |
1.066uM |
View
|
5-hydroxytryptamine (serotonin) receptor 1A |
BW-723C86 |
Serotonin 5-HT1A |
86% |
1.1278uM |
.6445uM |
View
|
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 |
BUPROPION |
Dopamine Transporter |
86% |
1.0338uM |
.8214uM |
View
|
tachykinin receptor 2 |
4-NONYLPHENOL |
Tachykinin NK2 |
86% |
4.514uM |
1.505uM |
View
|
sodium channel, voltage-gated, type IV, beta |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel associated protein 1 |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel associated protein 2 |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type III, beta |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type I, alpha |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type IX, alpha |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type VII, alpha |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
amiloride-sensitive cation channel 5, intestinal |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type III, beta |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type VIII, alpha polypeptide |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type XI, alpha |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type I, beta |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type 10, alpha polypeptide |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type IV, alpha polypeptide |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type V, alpha polypeptide |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type II, beta |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, nonvoltage-gated 1 alpha |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, nonvoltage-gated 1 gamma |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, nonvoltage-gated 1 beta |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
sodium channel, voltage-gated, type 2, alpha 1 polypeptide |
THIORIDAZINE |
Sodium Channel, Site 2 |
86% |
2.056uM |
1.876uM |
View
|
calcium channel, voltage-dependent, beta 4 subunit |
FLUPHENAZINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
2.534uM |
2.464uM |
View
|
calcium channel, voltage-dependent, beta 3 subunit |
FLUPHENAZINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
2.534uM |
2.464uM |
View
|
calcium channel, voltage-dependent, beta 2 subunit |
FLUPHENAZINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
2.534uM |
2.464uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1S subunit |
FLUPHENAZINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
2.534uM |
2.464uM |
View
|
calcium channel, voltage-dependent, alpha 1F subunit |
FLUPHENAZINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
2.534uM |
2.464uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1D subunit |
FLUPHENAZINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
2.534uM |
2.464uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1C subunit |
FLUPHENAZINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
2.534uM |
2.464uM |
View
|
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
FLUPHENAZINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
2.534uM |
2.464uM |
View
|
calcium channel, voltage-dependent, beta 1 subunit |
FLUPHENAZINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
2.534uM |
2.464uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1E subunit |
FLUPHENAZINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
2.534uM |
2.464uM |
View
|
calcium channel, voltage-dependent, N type, alpha 1B subunit |
FLUPHENAZINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
2.534uM |
2.464uM |
View
|
calcium channel, voltage-dependent, alpha2/delta subunit 1 |
FLUPHENAZINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
2.534uM |
2.464uM |
View
|
adrenergic receptor, alpha 2a |
DOXEPIN |
Adrenergic alpha2A |
89% |
1.335uM |
.501uM |
View
|
histamine receptor H 2 |
HALOPERIDOL |
Histamine H2 |
89% |
1.166uM |
1.147uM |
View
|
adrenergic receptor, alpha 2b |
MONTELUKAST |
Adrenergic alpha2C |
89% |
5.279uM |
.767uM |
View
|
adrenergic receptor, alpha 2c (Non-specific probe) |
MONTELUKAST |
Adrenergic alpha2C |
89% |
5.279uM |
.767uM |
View
|
5-hydroxytryptamine (serotonin) receptor 2B |
CITALOPRAM |
Serotonin 5-HT2B |
89% |
1.839uM |
1.171uM |
View
|
cholinergic receptor, muscarinic 3 |
MIANSERIN |
Muscarinic M3 |
89% |
1.405uM |
.298uM |
View
|
cholinergic receptor, muscarinic 1 |
MIANSERIN |
Muscarinic M1 |
89% |
1.423uM |
.343uM |
View
|
mitogen activated protein kinase 14 |
MC 258717 |
Protein Serine/Threonine Kinase, p38alpha |
89% |
2.272uM |
NoneNone |
View
|
mitogen-activated protein kinase 14 |
MC 258717 |
Protein Serine/Threonine Kinase, p38alpha |
89% |
2.272uM |
NoneNone |
View
|
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) |
1-(2-METHOXYBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE |
CYP450-2C9 Inhibition |
89% |
2uM |
NoneNone |
View
|
cytochrome P450, family 2, subfamily C, polypeptide 9 |
1-(2-METHOXYBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE |
CYP450-2C9 Inhibition |
89% |
2uM |
NoneNone |
View
|
adrenergic receptor, alpha 2a |
1-NAPHTHYL ISOTHIOCYANATE |
Adrenergic alpha2A |
89% |
6.272uM |
2.352uM |
View
|
cholinergic receptor, muscarinic 4 |
QUINACRINE |
Muscarinic M4 |
89% |
1.983uM |
.277uM |
View
|
cholinergic receptor, muscarinic 4 |
KETOTIFEN |
Muscarinic M4 |
89% |
1.009uM |
.141uM |
View
|
adrenergic receptor, alpha 2a |
SELEGILINE |
Adrenergic alpha2A |
89% |
1.798uM |
.674uM |
View
|
monoamine oxidase A |
NABUMETONE |
Monoamine Oxidase MAOA |
89% |
.998uM |
NoneNone |
View
|
monoamine oxidase A |
NABUMETONE |
Monoamine Oxidase MAOA |
89% |
.998uM |
NoneNone |
View
|
adrenergic receptor, alpha 2a |
NORTRIPTYLINE |
Adrenergic alpha2A |
89% |
.732uM |
.275uM |
View
|
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 |
OLANZAPINE |
Serotonin Transporter |
89% |
1.033uM |
.549uM |
View
|
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 |
NORETHINDRONE |
Serotonin Transporter |
89% |
4.537uM |
2.411uM |
View
|
5-hydroxytryptamine (serotonin) receptor 1A |
NORTRIPTYLINE |
Serotonin 5-HT1A |
89% |
1.868uM |
1.068uM |
View
|
adrenergic receptor, alpha 2a |
OXYMETAZOLINE |
Imidazoline I2, Central |
89% |
.027uM |
.018uM |
View
|
adrenergic receptor, alpha 2c (Non-specific probe) |
OXYMETAZOLINE |
Imidazoline I2, Central |
89% |
.027uM |
.018uM |
View
|
dopamine receptor 2 |
EBASTINE |
Dopamine D2L |
89% |
1.1491uM |
.383uM |
View
|
A3 adenosine receptor |
EBASTINE |
Adenosine A3 |
89% |
3.1953uM |
1.8061uM |
View
|
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 4 |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
gamma-aminobutyric acid A receptor, gamma 1 |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
gamma-aminobutyric acid A receptor, pi |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
AT hook, DNA binding motif, containing 1 (DBSS) |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
gamma-aminobutyric acid A receptor, theta |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
gamma-aminobutyric acid A receptor, gamma 2 |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 6 |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 5 |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
gamma-aminobutyric acid A receptor, alpha 2 |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
gamma-aminobutyric acid A receptor, alpha 1 |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 2 |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 1 |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
gamma-aminobutyric acid A receptor, delta |
CHLORDIAZEPOXIDE |
GABAA, Benzodiazepine, Central |
89% |
1.429uM |
1.164uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1S subunit |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, alpha 1F subunit |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1D subunit |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1C subunit |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, beta 1 subunit |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1E subunit |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, N type, alpha 1B subunit |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
calcium channel, voltage-dependent, alpha2/delta subunit 1 |
DICYCLOMINE |
Calcium Channel Type L, Benzothiazepine |
88% |
1.736uM |
1.543uM |
View
|
3-hydroxy-3-methylglutaryl-Coenzyme A reductase |
CISAPRIDE |
HMG-CoA Reductase |
88% |
3.37uM |
NoneNone |
View
|
3-hydroxy-3-methylglutaryl-Coenzyme A reductase |
CISAPRIDE |
HMG-CoA Reductase |
88% |
3.37uM |
NoneNone |
View
|
dopamine receptor 2 |
CISAPRIDE |
Dopamine D2L |
88% |
.473uM |
.158uM |
View
|
dopamine receptor D1A |
CARVEDILOL |
Dopamine D1 |
88% |
1.498uM |
.749uM |
View
|
adrenergic receptor, beta 3 |
TIMOLOL |
Adrenergic beta3 |
88% |
.452uM |
.339uM |
View
|
cholinergic receptor, muscarinic 5 |
FLUOXETINE |
Muscarinic M5 |
88% |
1.358uM |
.976uM |
View
|
phosphodiesterase 3B |
CILOSTAZOL |
Phosphodiesterase PDE3 |
88% |
.271uM |
NoneNone |
View
|
phosphodiesterase 3A |
CILOSTAZOL |
Phosphodiesterase PDE3 |
88% |
.271uM |
NoneNone |
View
|
adrenergic receptor, alpha 2b |
TICLOPIDINE |
Adrenergic alpha2C |
88% |
1.175uM |
.171uM |
View
|
adrenergic receptor, alpha 2c (Non-specific probe) |
TICLOPIDINE |
Adrenergic alpha2C |
88% |
1.175uM |
.171uM |
View
|
A3 adenosine receptor |
SULINDAC SULFIDE |
Adenosine A3 |
88% |
7.231uM |
4.087uM |
View
|
prostaglandin-endoperoxide synthase 1 |
MONOBENZONE |
Cyclooxygenase COX-1 |
88% |
1.019uM |
NoneNone |
View
|
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) |
MONOBENZONE |
Cyclooxygenase COX-1 |
88% |
1.019uM |
NoneNone |
View
|
calcium channel, voltage-dependent, beta 4 subunit |
HALOPERIDOL |
Calcium Channel Type L, Phenylalkylamine |
88% |
.552uM |
.536uM |
View
|
sodium channel, voltage-gated, type IX, alpha |
BENZTROPINE |
Sodium Channel, Site 2 |
88% |
1.68uM |
1.533uM |
View
|
adrenergic receptor, beta 1 |
LISURIDE |
Adrenergic beta1 |
88% |
.559uM |
.323uM |
View
|
adrenergic, beta-1-, receptor |
LISURIDE |
Adrenergic beta1 |
88% |
.559uM |
.323uM |
View
|
adrenergic receptor, alpha 2b |
MAPROTILINE |
Adrenergic alpha2C |
88% |
3.044uM |
.442uM |
View
|
adrenergic receptor, alpha 2c (Non-specific probe) |
MAPROTILINE |
Adrenergic alpha2C |
88% |
3.044uM |
.442uM |
View
|
dopamine receptor D1A |
IVERMECTIN |
Dopamine D1 |
88% |
4.5148uM |
2.2574uM |
View
|
5-hydroxytryptamine (serotonin) receptor 2C |
PYRILAMINE |
Serotonin 5-HT2C |
88% |
1.13uM |
.592uM |
View
|
mitogen activated protein kinase 14 |
VX-745 |
Protein Serine/Threonine Kinase, p38alpha |
88% |
.643uM |
NoneNone |
View
|
mitogen-activated protein kinase 14 |
VX-745 |
Protein Serine/Threonine Kinase, p38alpha |
88% |
.643uM |
NoneNone |
View
|
adrenergic receptor, alpha 1b |
ROXITHROMYCIN |
Adrenergic alpha1B |
88% |
.989uM |
.548uM |
View
|
adenosine A2a receptor |
SILDENAFIL |
Adenosine A2A |
88% |
.253uM |
.142uM |
View
|