Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
cytochrome P450, family 2, subfamily C, polypeptide 9 CLOSANTEL CYP450-2C9 Inhibition 89% 2uM NoneNone View
Cytochrom P450-2C19 monooxygenase MOSAPRIDE CYP450-2C19 Inhibition 89% 1uM NoneNone View
cholinergic receptor, muscarinic 5 DIPHENIDOL Muscarinic M5 89% 1.191uM .855uM View
thromboxane A synthase 1 BITHIONOL Thromboxane Synthetase 89% 1.84uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) BITHIONOL Thromboxane Synthetase 89% 1.84uM NoneNone View
adrenergic receptor, alpha 2a AMITRAZ Adrenergic alpha2A 89% .9269uM .3476uM View
FMS-like tyrosine kinase 1 DIGITONIN Vascular Endothelinal Growth Factor (VEGF) 89% 3.859uM 1.001uM View
fms-related tyrosine kinase 1 (vascular endothelial growth factor/vascular permeability factor receptor) DIGITONIN Vascular Endothelinal Growth Factor (VEGF) 89% 3.859uM 1.001uM View
adrenergic receptor, alpha 2a DIHYDROERGOCRISTINE MESYLATE Imidazoline I2, Central 89% .005428uM .003619uM View
adrenergic receptor, alpha 2c (Non-specific probe) DIHYDROERGOCRISTINE MESYLATE Imidazoline I2, Central 89% .005428uM .003619uM View
adrenergic receptor, alpha 1b EPINEPHRINE Adrenergic alpha1B 89% 1.766uM .977uM View
mu-opioid receptor MOR NELFINAVIR Opiate mu 89% 14.432uM 5.859uM View
adrenergic receptor, alpha 1b CINNARIZINE Adrenergic alpha1B 89% .906uM .502uM View
5-hydroxytryptamine receptor 6 SULFADIMETHOXINE Serotonin 5-HT6 87% 1.339uM .622uM View
Cytochrom P450-1A2 monooxygenase PROCHLORPERAZINE CYP450-1A2 Inhibition 87% 2uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 1A SAQUINAVIR Serotonin 5-HT1A 87% 4.273uM 2.442uM View
adrenergic receptor, alpha 2a SELEGILINE Imidazoline I2, Central 87% 1.614uM 1.076uM View
adrenergic receptor, alpha 2c (Non-specific probe) SELEGILINE Imidazoline I2, Central 87% 1.614uM 1.076uM View
adrenergic receptor, beta 3 OXICONAZOLE Adrenergic beta3 87% 4.7449uM 3.5587uM View
dopamine receptor D1A EBASTINE Dopamine D1 87% 1.1929uM .5965uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 MONTELUKAST Adrenergic, Norepinephrine Transporter 87% 2.689uM 2.667uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 RESVERATROL Adrenergic, Norepinephrine Transporter 87% 2.312uM 2.293uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 CETYLPYRIDINIUM BROMIDE Adrenergic, Norepinephrine Transporter 87% 2.653uM 2.631uM View
opioid receptor, sigma 1 RALOXIFENE Sigma1 87% .681uM .286uM View
5-hydroxytryptamine (serotonin) receptor 1B RALOXIFENE Serotonin 5-HT1B 87% 1.861uM .846uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 SIBUTRAMINE Dopamine Transporter 87% .632uM .502uM View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) STANOZOLOL CYP450-2C9 Inhibition 87% 1.1276uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 STANOZOLOL CYP450-2C9 Inhibition 87% 1.1276uM NoneNone View
adrenergic receptor, alpha 2b BENZETHONIUM CHLORIDE Adrenergic alpha2B 87% .643uM .294uM View
cholinergic receptor, muscarinic 5 BENZETHONIUM CHLORIDE Muscarinic M5 87% .134uM .096uM View
5-hydroxytryptamine (serotonin) receptor 1A ASTEMIZOLE Serotonin 5-HT1A 87% .767uM .438uM View
nuclear receptor subfamily 3, group C, member 1 SPIRONOLACTONE Glucocorticoid 87% 1.9025uM .8648uM View
dopamine receptor D3 BAY 11-7085 Dopamine D3 87% 3.46uM 1.175uM View
5-hydroxytryptamine receptor 6 ASTEMIZOLE Serotonin 5-HT6 87% 3.266uM 1.516uM View
Sigma-2 Receptor CLOMIPHENE Sigma2 87% .049uM .03uM View
mitogen activated protein kinase 1 ANTIMYCIN A Protein Serine/Threonine Kinase, ERK2 87% 2.116uM NoneNone View
mitogen-activated protein kinase 1 ANTIMYCIN A Protein Serine/Threonine Kinase, ERK2 87% 2.116uM NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, gamma subunit 8 NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, gamma subunit 7 NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
calcium channel, voltage-dependent, gamma subunit 6 NELFINAVIR Calcium Channel Type L, Dihydropyridine 87% 9.84uM 6.324uM View
Sigma-2 Receptor TERBINAFINE Sigma2 87% .0354uM .0218uM View
adrenergic receptor, alpha 1d (Non-specific probe) CINNARIZINE Adrenergic alpha1D 87% 1.167uM .573uM View
calcium channel, voltage-dependent, gamma subunit 3 PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, gamma subunit 2 PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, gamma subunit 1 PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, beta 4 subunit PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, beta 3 subunit PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, beta 2 subunit PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, alpha 1F subunit PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, beta 1 subunit PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, gamma subunit 8 PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, gamma subunit 7 PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, gamma subunit 6 PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, gamma subunit 5 PAROXETINE Calcium Channel Type L, Dihydropyridine 87% 1.476uM .949uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 U-78517F Calcium Channel Type L, Dihydropyridine 86% 1.659uM 1.066uM View
mitogen activated protein kinase 14 U-78517F Protein Serine/Threonine Kinase, p38alpha 86% 5.596uM NoneNone View
mitogen-activated protein kinase 14 U-78517F Protein Serine/Threonine Kinase, p38alpha 86% 5.596uM NoneNone View
cholinergic receptor, muscarinic 3 AMOXAPINE Muscarinic M3 86% 1.781uM .378uM View
melanocortin 4 receptor AMIODARONE Melanocortin MC4 86% 13.755uM 13.226uM View
cholinergic receptor, muscarinic 1 AMIODARONE Muscarinic M1 86% 2.613uM .629uM View
epidermal growth factor receptor TAMOXIFEN Protein Tyrosine Kinase, EGF Receptor 86% 3.553uM NoneNone View
dopamine receptor D3 DICYCLOMINE Dopamine D3 86% 1.21uM .411uM View
adrenergic receptor, alpha 1d (Non-specific probe) CISAPRIDE Adrenergic alpha1D 86% .189uM .093uM View
calcium channel, voltage-dependent, gamma subunit 8 CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, gamma subunit 7 CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, gamma subunit 6 CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, gamma subunit 5 CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, gamma subunit 4 CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, gamma subunit 3 CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, gamma subunit 2 CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, gamma subunit 1 CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, beta 4 subunit CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, beta 3 subunit CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, beta 2 subunit CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, alpha 1F subunit CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, beta 1 subunit CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 CLOMIPRAMINE Calcium Channel Type L, Phenylalkylamine 86% .506uM .492uM View
5-hydroxytryptamine (serotonin) receptor 5B CARVEDILOL Serotonin 5-HT4 86% 1.088uM .181uM View
5-hydroxytryptamine (serotonin) receptor 4 CARVEDILOL Serotonin 5-HT4 86% 1.088uM .181uM View
calcium channel, voltage-dependent, gamma subunit 8 CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, gamma subunit 7 CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, gamma subunit 6 CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, gamma subunit 5 CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, gamma subunit 4 CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, gamma subunit 3 CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, gamma subunit 2 CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, gamma subunit 1 CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, beta 4 subunit CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, beta 3 subunit CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, beta 2 subunit CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, alpha 1F subunit CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CLOZAPINE Calcium Channel Type L, Benzothiazepine 86% 3.752uM 3.335uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit FLUNARIZINE Calcium Channel Type L, Dihydropyridine 90% 1.012uM .65uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit FLUNARIZINE Calcium Channel Type L, Dihydropyridine 90% 1.012uM .65uM View
calcium channel, voltage-dependent, beta 1 subunit FLUNARIZINE Calcium Channel Type L, Dihydropyridine 90% 1.012uM .65uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit FLUNARIZINE Calcium Channel Type L, Dihydropyridine 90% 1.012uM .65uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit FLUNARIZINE Calcium Channel Type L, Dihydropyridine 90% 1.012uM .65uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 FLUNARIZINE Calcium Channel Type L, Dihydropyridine 90% 1.012uM .65uM View
Cytochrom P450-2D6 monooxygenase TICLOPIDINE CYP450-2D6 Inhibition 90% 6.2928uM NoneNone View
Cytochrom P450-2D6 monooxygenase YOHIMBINE CYP450-2D6 Inhibition 90% 2.0317uM NoneNone View
Cytochrom P450-2D6 monooxygenase PHENTOLAMINE CYP450-2D6 Inhibition 90% 10uM NoneNone View
Cytochrom P450-2D6 monooxygenase PYRILAMINE CYP450-2D6 Inhibition 90% .3uM NoneNone View
Cytochrom P450-2D6 monooxygenase CISAPRIDE CYP450-2D6 Inhibition 90% .07uM NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) FELODIPINE CYP450-2C9 Inhibition 90% 4.5795uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 FELODIPINE CYP450-2C9 Inhibition 90% 4.5795uM NoneNone View
mitogen activated protein kinase 1 3,3',4',5-TETRACHLOROSALICYLANILIDE Protein Serine/Threonine Kinase, ERK2 90% .886uM NoneNone View
mitogen-activated protein kinase 1 3,3',4',5-TETRACHLOROSALICYLANILIDE Protein Serine/Threonine Kinase, ERK2 90% .886uM NoneNone View
adenosine A2a receptor BITHIONOL Adenosine A2A 90% 1.167uM .655uM View
A3 adenosine receptor CLOSANTEL Adenosine A3 90% .096uM .054uM View
acetylcholinesterase (YT blood group) CLOSANTEL Acetylcholinesterase 90% 2.951uM NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase CLOSANTEL Acetylcholinesterase 90% 2.951uM NoneNone View
acetylcholinesterase CLOSANTEL Acetylcholinesterase 90% 2.951uM NoneNone View
Protein-tyrosine kinase, Fyn GRAMICIDIN Protein Tyrosine Kinase, Fyn 90% 3.331uM NoneNone View
adrenergic receptor, alpha 2a CINNARIZINE Adrenergic alpha2A 90% .444uM .167uM View
5-hydroxytryptamine (serotonin) receptor 2B BUSPIRONE Serotonin 5-HT2B 90% .75uM .477uM View
5-hydroxytryptamine (serotonin) receptor 1A QUETIAPINE Serotonin 5-HT1A 90% 1.4264uM .8151uM View
mu-opioid receptor MOR DIHYDROERGOCRISTINE MESYLATE Opiate mu 90% .85uM .345uM View
5-hydroxytryptamine (serotonin) receptor 2A PYRILAMINE Serotonin 5-HT2A 90% .997uM .285uM View
dopamine receptor 2 PROMAZINE Dopamine D2L 90% .505uM .168uM View
adrenergic receptor, alpha 2a TERCONAZOLE Imidazoline I2, Central 90% 2.226uM 1.484uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 3 CHLORDIAZEPOXIDE GABAA, Benzodiazepine, Central 89% 1.429uM 1.164uM View
calcium channel, voltage-dependent, beta 2 subunit PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, alpha 1F subunit PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, beta 1 subunit PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, gamma subunit 8 PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, gamma subunit 7 PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, gamma subunit 6 PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, gamma subunit 5 PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, gamma subunit 4 PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, gamma subunit 3 PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, gamma subunit 2 PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, gamma subunit 1 PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, beta 4 subunit PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
calcium channel, voltage-dependent, beta 3 subunit PROMETHAZINE Calcium Channel Type L, Phenylalkylamine 89% .866uM .842uM View
A3 adenosine receptor LACIDIPINE Adenosine A3 89% 4.036uM 2.281uM View
calcium channel, voltage-dependent, beta 3 subunit HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, beta 2 subunit HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, alpha 1F subunit HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, beta 1 subunit HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, gamma subunit 8 HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, gamma subunit 7 HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, gamma subunit 6 HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, gamma subunit 5 HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, gamma subunit 4 HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, gamma subunit 3 HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, gamma subunit 2 HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
calcium channel, voltage-dependent, gamma subunit 1 HALOPERIDOL Calcium Channel Type L, Phenylalkylamine 88% .552uM .536uM View
Protein-tyrosine kinase, Fyn GENTIAN VIOLET Protein Tyrosine Kinase, Fyn 88% 2.148uM NoneNone View
opioid receptor, sigma 1 MEPAZINE Sigma1 88% .18uM .076uM View
dopamine receptor D3 LOPERAMIDE Dopamine D3 88% 1.337uM .454uM View
opioid receptor, delta 1 LOPERAMIDE Opiate delta 88% .896uM .316uM View
dopamine receptor D1A METHYSERGIDE Dopamine D1 88% .943uM .472uM View
arachidonate 15-lipoxygenase, second type MITOXANTRONE Lipoxygenase 15-LO 88% 1.7853uM NoneNone View
arachidonate 15-lipoxygenase MITOXANTRONE Lipoxygenase 15-LO 88% 1.7853uM NoneNone View
arachidonate 15-lipoxygenase MITOXANTRONE Lipoxygenase 15-LO 88% 1.7853uM NoneNone View
epidermal growth factor receptor L-744832 Protein Tyrosine Kinase, EGF Receptor 88% 3.216uM NoneNone View
matrix metalloproteinase 1 (interstitial collagenase) IRINOTECAN Protease, Matrix Metalloprotease-1 (MMP-1) 88% 6.06uM NoneNone View
5-hydroxytryptamine receptor 6 KETOTIFEN Serotonin 5-HT6 88% 1.141uM .53uM View
adrenergic receptor, alpha 2a KETOTIFEN Adrenergic alpha2A 88% 2.187uM .82uM View
thromboxane A synthase 1 RITONAVIR Thromboxane Synthetase 88% .076uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) RITONAVIR Thromboxane Synthetase 88% .076uM NoneNone View
adrenergic receptor, beta 3 MONTELUKAST Adrenergic beta3 88% 4.3uM 3.2uM View
phosphodiesterase 4A, cAMP specific PAPAVERINE Phosphodiesterase PDE4 88% .817uM NoneNone View
phosphodiesterase 4C, cAMP-specific PAPAVERINE Phosphodiesterase PDE4 88% .817uM NoneNone View
phosphodiesterase 4D PAPAVERINE Phosphodiesterase PDE4 88% .817uM NoneNone View
phosphodiesterase 4B, cAMP specific PAPAVERINE Phosphodiesterase PDE4 88% .817uM NoneNone View
phosphodiesterase 3B PAPAVERINE Phosphodiesterase PDE3 88% .665uM NoneNone View
phosphodiesterase 3A PAPAVERINE Phosphodiesterase PDE3 88% .665uM NoneNone View