5-hydroxytryptamine (serotonin) receptor 2A |
GUANFACINE |
Serotonin 5-HT2A |
75% |
3.014uM |
.861uM |
View
|
potassium voltage-gated channel, subfamily H (eag-related), member 1 |
FLUPHENAZINE |
Potassium Channel HERG |
75% |
5.7058uM |
4.6746uM |
View
|
potassium voltage-gated channel, subfamily H (eag-related), member 1 |
FLUPHENAZINE |
Potassium Channel HERG |
75% |
5.7058uM |
4.6746uM |
View
|
potassium voltage-gated channel, subfamily H, member 8 |
FLUPHENAZINE |
Potassium Channel HERG |
75% |
5.7058uM |
4.6746uM |
View
|
potassium voltage-gated channel, subfamily H (eag-related), member 6 |
FLUPHENAZINE |
Potassium Channel HERG |
75% |
5.7058uM |
4.6746uM |
View
|
potassium voltage-gated channel, subfamily H (eag-related), member 7 |
FLUPHENAZINE |
Potassium Channel HERG |
75% |
5.7058uM |
4.6746uM |
View
|
potassium voltage-gated channel, subfamily H (eag-related), member 2 |
FLUPHENAZINE |
Potassium Channel HERG |
75% |
5.7058uM |
4.6746uM |
View
|
potassium voltage-gated channel, subfamily H (eag-related), member 5 |
FLUPHENAZINE |
Potassium Channel HERG |
75% |
5.7058uM |
4.6746uM |
View
|
potassium voltage-gated channel, subfamily H (eag-related), member 3 |
FLUPHENAZINE |
Potassium Channel HERG |
75% |
5.7058uM |
4.6746uM |
View
|
potassium voltage-gated channel, subfamily H (eag-related), member 4 |
FLUPHENAZINE |
Potassium Channel HERG |
75% |
5.7058uM |
4.6746uM |
View
|
cholinergic receptor, muscarinic 5 |
TRANS-PLATINUM(II)DIAMMINE DICHLORIDE |
Muscarinic M5 |
75% |
5.9254uM |
4.2571uM |
View
|
Cytochrom P450-2D6 monooxygenase |
METHAPYRILENE |
CYP450-2D6 Inhibition |
75% |
2.7564uM |
NoneNone |
View
|
Cytochrom P450-1A2 monooxygenase |
PROPAFENONE |
CYP450-1A2 Inhibition |
75% |
3.292uM |
NoneNone |
View
|
adrenergic receptor, beta 3 |
SULOCTIDIL |
Adrenergic beta3 |
75% |
4.9963uM |
3.7472uM |
View
|
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 |
LEVOBUNOLOL |
Serotonin Transporter |
75% |
4.898uM |
2.602uM |
View
|
5-hydroxytryptamine (serotonin) receptor 2B |
DIMENHYDRINATE |
Serotonin 5-HT2B |
75% |
1.724uM |
1.097uM |
View
|
mitogen activated protein kinase 14 |
MONTELUKAST |
Protein Serine/Threonine Kinase, p38alpha |
75% |
.856uM |
NoneNone |
View
|
mitogen-activated protein kinase 14 |
MONTELUKAST |
Protein Serine/Threonine Kinase, p38alpha |
75% |
.856uM |
NoneNone |
View
|
platelet-activating factor receptor |
CILOSTAMIDE |
Platelet Activating Factor (PAF) |
75% |
3.687uM |
1.917uM |
View
|
cholinergic receptor, muscarinic 4 |
FLUNARIZINE |
Muscarinic M4 |
75% |
5.656uM |
.789uM |
View
|
dopamine receptor D4 |
THIORIDAZINE |
Dopamine D4.2 |
75% |
1.468uM |
.515uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1E subunit |
SPIRADOLINE |
Calcium Channel Type L, Phenylalkylamine |
78% |
5.24uM |
5.095uM |
View
|
calcium channel, voltage-dependent, N type, alpha 1B subunit |
SPIRADOLINE |
Calcium Channel Type L, Phenylalkylamine |
78% |
5.24uM |
5.095uM |
View
|
calcium channel, voltage-dependent, alpha2/delta subunit 1 |
SPIRADOLINE |
Calcium Channel Type L, Phenylalkylamine |
78% |
5.24uM |
5.095uM |
View
|
acetylcholinesterase (YT blood group) |
BUTENAFINE |
Acetylcholinesterase |
78% |
6.9071uM |
NoneNone |
View
|
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase |
BUTENAFINE |
Acetylcholinesterase |
78% |
6.9071uM |
NoneNone |
View
|
acetylcholinesterase |
BUTENAFINE |
Acetylcholinesterase |
78% |
6.9071uM |
NoneNone |
View
|
cholinergic receptor, muscarinic 1 |
QUETIAPINE |
Muscarinic M1 |
78% |
2.615uM |
.6298uM |
View
|
A3 adenosine receptor |
VX-745 |
Adenosine A3 |
78% |
8.547uM |
4.831uM |
View
|
dopamine receptor D3 |
TERCONAZOLE |
Dopamine D3 |
78% |
4.712uM |
1.6uM |
View
|
adrenergic receptor, alpha 2a |
SEMUSTINE |
Adrenergic alpha2A |
78% |
4.809uM |
1.803uM |
View
|
histamine receptor H 1 |
METERGOLINE |
Histamine H1, Central |
78% |
4.133uM |
.48uM |
View
|
cholinergic receptor, muscarinic 5 |
PENTAMIDINE |
Muscarinic M5 |
78% |
2.885uM |
2.073uM |
View
|
5-hydroxytryptamine (serotonin) receptor 2C |
PENTAMIDINE |
Serotonin 5-HT2C |
78% |
3.278uM |
1.717uM |
View
|
adrenergic receptor, alpha 2a |
PRAZOSIN |
Imidazoline I2, Central |
78% |
.949uM |
.633uM |
View
|
adrenergic receptor, alpha 2c (Non-specific probe) |
PRAZOSIN |
Imidazoline I2, Central |
78% |
.949uM |
.633uM |
View
|
Protein-tyrosine kinase, Fyn |
PROCHLORPERAZINE |
Protein Tyrosine Kinase, Fyn |
78% |
5.684uM |
NoneNone |
View
|
calcium channel, voltage-dependent, gamma subunit 8 |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, gamma subunit 7 |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, gamma subunit 6 |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, gamma subunit 5 |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, gamma subunit 4 |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, gamma subunit 3 |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, gamma subunit 2 |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, gamma subunit 1 |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, beta 4 subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, beta 3 subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, beta 2 subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1S subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, alpha 1F subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1D subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1C subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
calcium channel, voltage-dependent, beta 1 subunit |
PERGOLIDE |
Calcium Channel Type L, Benzothiazepine |
78% |
3.301uM |
2.934uM |
View
|
Cytochrom P450-2C19 monooxygenase |
ROTENONE |
CYP450-2C19 Inhibition |
78% |
3.6486uM |
NoneNone |
View
|
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 |
BW-723C86 |
Adrenergic, Norepinephrine Transporter |
78% |
3.6257uM |
3.5957uM |
View
|
Cytochrom P450-2D6 monooxygenase |
CYCLIZINE |
CYP450-2D6 Inhibition |
78% |
6.2175uM |
NoneNone |
View
|
epidermal growth factor receptor |
THIORIDAZINE |
Protein Tyrosine Kinase, EGF Receptor |
78% |
2.947uM |
NoneNone |
View
|
mitogen activated protein kinase 14 |
ZAFIRLUKAST |
Protein Serine/Threonine Kinase, p38alpha |
78% |
.353uM |
NoneNone |
View
|
mitogen-activated protein kinase 14 |
ZAFIRLUKAST |
Protein Serine/Threonine Kinase, p38alpha |
78% |
.353uM |
NoneNone |
View
|
cholinergic receptor, muscarinic 3 |
MONTELUKAST |
Muscarinic M3 |
78% |
6.626uM |
1.404uM |
View
|
cannabinoid receptor 1 (brain) |
FLUNARIZINE |
Cannabinoid CB1 |
78% |
3.028uM |
2.391uM |
View
|
calcium channel, voltage-dependent, gamma subunit 8 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
calcium channel, voltage-dependent, gamma subunit 7 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
calcium channel, voltage-dependent, gamma subunit 6 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
calcium channel, voltage-dependent, gamma subunit 5 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
calcium channel, voltage-dependent, gamma subunit 4 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
calcium channel, voltage-dependent, gamma subunit 3 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
calcium channel, voltage-dependent, gamma subunit 2 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
calcium channel, voltage-dependent, gamma subunit 1 |
DIMENHYDRINATE |
Calcium Channel Type L, Phenylalkylamine |
78% |
3.344uM |
3.251uM |
View
|
sodium channel, voltage-gated, type III, beta |
PROMAZINE |
Sodium Channel, Site 2 |
77% |
2.573uM |
2.347uM |
View
|
sodium channel, voltage-gated, type VIII, alpha polypeptide |
PROMAZINE |
Sodium Channel, Site 2 |
77% |
2.573uM |
2.347uM |
View
|
5-hydroxytryptamine (serotonin) receptor 2C |
TERCONAZOLE |
Serotonin 5-HT2C |
77% |
6.961uM |
3.646uM |
View
|
adrenergic receptor, alpha 1d (Non-specific probe) |
TERCONAZOLE |
Adrenergic alpha1D |
77% |
14.385uM |
7.07uM |
View
|
cholinergic receptor, muscarinic 2 |
PROCHLORPERAZINE |
Muscarinic M2 |
77% |
3.112uM |
1.107uM |
View
|
A3 adenosine receptor |
TROGLITAZONE |
Adenosine A3 |
77% |
5.208uM |
2.943uM |
View
|
adrenergic receptor, alpha 1d (Non-specific probe) |
ECONAZOLE |
Adrenergic alpha1D |
77% |
8.897uM |
4.373uM |
View
|
calcium channel, voltage-dependent, gamma subunit 8 |
SULCONAZOLE |
Calcium Channel Type L, Dihydropyridine |
77% |
2.427uM |
1.56uM |
View
|
calcium channel, voltage-dependent, gamma subunit 7 |
SULCONAZOLE |
Calcium Channel Type L, Dihydropyridine |
77% |
2.427uM |
1.56uM |
View
|
calcium channel, voltage-dependent, gamma subunit 6 |
SULCONAZOLE |
Calcium Channel Type L, Dihydropyridine |
77% |
2.427uM |
1.56uM |
View
|
calcium channel, voltage-dependent, gamma subunit 5 |
SULCONAZOLE |
Calcium Channel Type L, Dihydropyridine |
77% |
2.427uM |
1.56uM |
View
|
calcium channel, voltage-dependent, gamma subunit 4 |
SULCONAZOLE |
Calcium Channel Type L, Dihydropyridine |
77% |
2.427uM |
1.56uM |
View
|
Protein-tyrosine kinase, Fyn |
BETA-NAPHTHOFLAVONE |
Protein Tyrosine Kinase, Fyn |
77% |
2.5149uM |
NoneNone |
View
|
epidermal growth factor receptor |
PERHEXILINE |
Protein Tyrosine Kinase, EGF Receptor |
77% |
1.4852uM |
NoneNone |
View
|
Cytochrom P450-2C19 monooxygenase |
BUPROPION |
CYP450-2C19 Inhibition |
77% |
1.9983uM |
NoneNone |
View
|
5-hydroxytryptamine receptor 6 |
PROPAFENONE |
Serotonin 5-HT6 |
77% |
1.863uM |
.865uM |
View
|
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 |
AMBROXOL |
Serotonin Transporter |
77% |
3.391uM |
1.802uM |
View
|
Protein-tyrosine kinase, Fyn |
TERFENADINE |
Protein Tyrosine Kinase, Fyn |
77% |
6.123uM |
NoneNone |
View
|
mu-opioid receptor MOR |
DOMPERIDONE |
Opiate mu |
77% |
4.218uM |
1.712uM |
View
|
histamine receptor H 2 |
IMATINIB |
Histamine H2 |
77% |
1.963uM |
1.93uM |
View
|
dopamine receptor D3 |
CYCLIZINE |
Dopamine D3 |
77% |
2.992uM |
1.016uM |
View
|
Cytochrom P450-2D6 monooxygenase |
LOPERAMIDE |
CYP450-2D6 Inhibition |
77% |
2uM |
NoneNone |
View
|
Cytochrom P450-2C19 monooxygenase |
ETHYLESTRENOL |
CYP450-2C19 Inhibition |
77% |
1.2907uM |
NoneNone |
View
|
Cytochrom P450-2C19 monooxygenase |
RAPAMYCIN |
CYP450-2C19 Inhibition |
77% |
4uM |
NoneNone |
View
|
Cytochrom P450-2C19 monooxygenase |
RESVERATROL |
CYP450-2C19 Inhibition |
77% |
3uM |
NoneNone |
View
|
A3 adenosine receptor |
HYDROXYPROGESTERONE |
Adenosine A3 |
77% |
4.73uM |
2.674uM |
View
|
5-hydroxytryptamine (serotonin) receptor 2A |
DIPHENIDOL |
Serotonin 5-HT2A |
77% |
2.586uM |
.739uM |
View
|
estrogen receptor 1 |
ETHYLESTRENOL |
Estrogen ERalpha |
77% |
1.121uM |
.32uM |
View
|
estrogen receptor 1 |
ETHYLESTRENOL |
Estrogen ERalpha |
77% |
1.121uM |
.32uM |
View
|
adrenergic receptor, alpha 2a |
MOXONIDINE |
Imidazoline I2, Central |
77% |
1.4764uM |
.9843uM |
View
|
adrenergic receptor, alpha 2c (Non-specific probe) |
MOXONIDINE |
Imidazoline I2, Central |
77% |
1.4764uM |
.9843uM |
View
|
Protein-tyrosine kinase, Fyn |
METHYLDOPA |
Protein Tyrosine Kinase, Fyn |
77% |
5.176uM |
NoneNone |
View
|
calcium channel, voltage-dependent, gamma subunit 8 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, gamma subunit 7 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, gamma subunit 6 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, gamma subunit 5 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, gamma subunit 4 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, gamma subunit 3 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, gamma subunit 2 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, gamma subunit 1 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, beta 4 subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, beta 3 subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, beta 2 subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1S subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, alpha 1F subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1D subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1C subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, beta 1 subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1E subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, N type, alpha 1B subunit |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
calcium channel, voltage-dependent, alpha2/delta subunit 1 |
LISURIDE |
Calcium Channel Type L, Benzothiazepine |
77% |
3.522uM |
3.131uM |
View
|
epidermal growth factor receptor |
TERFENADINE |
Protein Tyrosine Kinase, EGF Receptor |
76% |
3.566uM |
NoneNone |
View
|
epidermal growth factor receptor |
ZAFIRLUKAST |
Protein Tyrosine Kinase, EGF Receptor |
76% |
5.751uM |
NoneNone |
View
|
angiotensin 1 converting enzyme 1 |
IODOQUINOL |
Protease, Angiotensin Converting Enzyme |
76% |
.906uM |
NoneNone |
View
|
angiotensin I converting enzyme (peptidyl-dipeptidase A) 1 |
IODOQUINOL |
Protease, Angiotensin Converting Enzyme |
76% |
.906uM |
NoneNone |
View
|
nitric oxide synthase 3 (endothelial cell) |
CHLORZOXAZONE |
Nitric Oxide Synthase, Constitutive (cNOS) |
76% |
2.794uM |
NoneNone |
View
|
nitric oxide synthase 3, endothelial cell |
CHLORZOXAZONE |
Nitric Oxide Synthase, Constitutive (cNOS) |
76% |
2.794uM |
NoneNone |
View
|
cholinergic receptor, muscarinic 4 |
CINNARIZINE |
Muscarinic M4 |
76% |
3.66uM |
.51uM |
View
|
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) |
ALPHA-ERGOCRYPTINE |
CYP450-2C9 Inhibition |
76% |
6uM |
NoneNone |
View
|
cytochrome P450, family 2, subfamily C, polypeptide 9 |
ALPHA-ERGOCRYPTINE |
CYP450-2C9 Inhibition |
76% |
6uM |
NoneNone |
View
|
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) |
RWJ-68354 |
CYP450-2C9 Inhibition |
76% |
1uM |
NoneNone |
View
|
cytochrome P450, family 2, subfamily C, polypeptide 9 |
RWJ-68354 |
CYP450-2C9 Inhibition |
76% |
1uM |
NoneNone |
View
|
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) |
PHENYLHYDRAZINE |
CYP450-2C9 Inhibition |
76% |
6uM |
NoneNone |
View
|
cytochrome P450, family 2, subfamily C, polypeptide 9 |
PHENYLHYDRAZINE |
CYP450-2C9 Inhibition |
76% |
6uM |
NoneNone |
View
|
Cytochrom P450-2C19 monooxygenase |
NOSCAPINE |
CYP450-2C19 Inhibition |
76% |
.4003uM |
NoneNone |
View
|
adrenergic receptor, alpha 2b |
BERBERINE CHLORIDE |
Adrenergic alpha2C |
76% |
2.837uM |
.412uM |
View
|
adrenergic receptor, alpha 2c (Non-specific probe) |
BERBERINE CHLORIDE |
Adrenergic alpha2C |
76% |
2.837uM |
.412uM |
View
|
phosphodiesterase 3B |
MILRINONE |
Phosphodiesterase PDE3 |
76% |
.9585uM |
NoneNone |
View
|
phosphodiesterase 3A |
MILRINONE |
Phosphodiesterase PDE3 |
76% |
.9585uM |
NoneNone |
View
|
melanocortin 5 receptor |
DIGITONIN |
Melanocortin MC5 |
76% |
3.88uM |
3.639uM |
View
|
sodium channel, voltage-gated, type IV, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel associated protein 1 |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel associated protein 2 |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type III, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type I, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type IX, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type VII, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
amiloride-sensitive cation channel 5, intestinal |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type III, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type VIII, alpha polypeptide |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type XI, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type I, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type 10, alpha polypeptide |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type IV, alpha polypeptide |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type V, alpha polypeptide |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type II, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, nonvoltage-gated 1 alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, nonvoltage-gated 1 gamma |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, nonvoltage-gated 1 beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type 2, alpha 1 polypeptide |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type XI, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, nonvoltage-gated 1, gamma |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, nonvoltage-gated 1, delta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, nonvoltage-gated 1 alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type X, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type IX, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage gated, type VIII, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type VII, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type IV, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type IV, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type III, alpha |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
sodium channel, voltage-gated, type II, beta |
MAPROTILINE |
Sodium Channel, Site 2 |
76% |
2.572uM |
2.346uM |
View
|
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 |
CLEMASTINE |
Dopamine Transporter |
89% |
.678uM |
.538uM |
View
|
adrenergic receptor, alpha 1d (Non-specific probe) |
CLEMASTINE |
Adrenergic alpha1D |
89% |
.032uM |
.015uM |
View
|
5-hydroxytryptamine (serotonin) receptor 1B |
CLEMASTINE |
Serotonin 5-HT1B |
89% |
.359uM |
.22uM |
View
|
calcium channel, voltage-dependent, gamma subunit 4 |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, gamma subunit 3 |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, gamma subunit 2 |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, gamma subunit 1 |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, beta 4 subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, beta 3 subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, beta 2 subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1S subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, alpha 1F subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1D subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1C subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, beta 1 subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
calcium channel, voltage-dependent, L type, alpha 1E subunit |
CLEMASTINE |
Calcium Channel Type L, Phenylalkylamine |
89% |
.508uM |
.493uM |
View
|
adrenergic receptor, alpha 2b |
DOMPERIDONE |
Adrenergic alpha2C |
89% |
1.011uM |
.147uM |
View
|
adrenergic receptor, alpha 2c (Non-specific probe) |
DOMPERIDONE |
Adrenergic alpha2C |
89% |
1.011uM |
.147uM |
View
|
cholinergic receptor, muscarinic 2 |
PENTAMIDINE |
Muscarinic M2 |
89% |
1.425uM |
.507uM |
View
|
adrenergic receptor, alpha 2b |
EPINEPHRINE |
Adrenergic alpha2B |
89% |
.869uM |
.397uM |
View
|
adrenergic receptor, alpha 2a |
METOCLOPRAMIDE |
Imidazoline I2, Central |
89% |
.708uM |
.472uM |
View
|
adrenergic receptor, alpha 2c (Non-specific probe) |
METOCLOPRAMIDE |
Imidazoline I2, Central |
89% |
.708uM |
.472uM |
View
|
calcium channel, voltage-dependent, gamma subunit 8 |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|
calcium channel, voltage-dependent, gamma subunit 7 |
MICONAZOLE |
Calcium Channel Type L, Phenylalkylamine |
89% |
3.788uM |
3.683uM |
View
|