Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
5-hydroxytryptamine (serotonin) receptor 2A GUANFACINE Serotonin 5-HT2A 75% 3.014uM .861uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H, member 8 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 6 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 7 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 2 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 5 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 3 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
potassium voltage-gated channel, subfamily H (eag-related), member 4 FLUPHENAZINE Potassium Channel HERG 75% 5.7058uM 4.6746uM View
cholinergic receptor, muscarinic 5 TRANS-PLATINUM(II)DIAMMINE DICHLORIDE Muscarinic M5 75% 5.9254uM 4.2571uM View
Cytochrom P450-2D6 monooxygenase METHAPYRILENE CYP450-2D6 Inhibition 75% 2.7564uM NoneNone View
Cytochrom P450-1A2 monooxygenase PROPAFENONE CYP450-1A2 Inhibition 75% 3.292uM NoneNone View
adrenergic receptor, beta 3 SULOCTIDIL Adrenergic beta3 75% 4.9963uM 3.7472uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 LEVOBUNOLOL Serotonin Transporter 75% 4.898uM 2.602uM View
5-hydroxytryptamine (serotonin) receptor 2B DIMENHYDRINATE Serotonin 5-HT2B 75% 1.724uM 1.097uM View
mitogen activated protein kinase 14 MONTELUKAST Protein Serine/Threonine Kinase, p38alpha 75% .856uM NoneNone View
mitogen-activated protein kinase 14 MONTELUKAST Protein Serine/Threonine Kinase, p38alpha 75% .856uM NoneNone View
platelet-activating factor receptor CILOSTAMIDE Platelet Activating Factor (PAF) 75% 3.687uM 1.917uM View
cholinergic receptor, muscarinic 4 FLUNARIZINE Muscarinic M4 75% 5.656uM .789uM View
dopamine receptor D4 THIORIDAZINE Dopamine D4.2 75% 1.468uM .515uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 SPIRADOLINE Calcium Channel Type L, Phenylalkylamine 78% 5.24uM 5.095uM View
acetylcholinesterase (YT blood group) BUTENAFINE Acetylcholinesterase 78% 6.9071uM NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase BUTENAFINE Acetylcholinesterase 78% 6.9071uM NoneNone View
acetylcholinesterase BUTENAFINE Acetylcholinesterase 78% 6.9071uM NoneNone View
cholinergic receptor, muscarinic 1 QUETIAPINE Muscarinic M1 78% 2.615uM .6298uM View
A3 adenosine receptor VX-745 Adenosine A3 78% 8.547uM 4.831uM View
dopamine receptor D3 TERCONAZOLE Dopamine D3 78% 4.712uM 1.6uM View
adrenergic receptor, alpha 2a SEMUSTINE Adrenergic alpha2A 78% 4.809uM 1.803uM View
histamine receptor H 1 METERGOLINE Histamine H1, Central 78% 4.133uM .48uM View
cholinergic receptor, muscarinic 5 PENTAMIDINE Muscarinic M5 78% 2.885uM 2.073uM View
5-hydroxytryptamine (serotonin) receptor 2C PENTAMIDINE Serotonin 5-HT2C 78% 3.278uM 1.717uM View
adrenergic receptor, alpha 2a PRAZOSIN Imidazoline I2, Central 78% .949uM .633uM View
adrenergic receptor, alpha 2c (Non-specific probe) PRAZOSIN Imidazoline I2, Central 78% .949uM .633uM View
Protein-tyrosine kinase, Fyn PROCHLORPERAZINE Protein Tyrosine Kinase, Fyn 78% 5.684uM NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, gamma subunit 7 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, gamma subunit 6 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, gamma subunit 5 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, gamma subunit 4 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, gamma subunit 3 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, gamma subunit 2 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, gamma subunit 1 PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, beta 4 subunit PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, beta 3 subunit PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, beta 2 subunit PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, alpha 1F subunit PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
calcium channel, voltage-dependent, beta 1 subunit PERGOLIDE Calcium Channel Type L, Benzothiazepine 78% 3.301uM 2.934uM View
Cytochrom P450-2C19 monooxygenase ROTENONE CYP450-2C19 Inhibition 78% 3.6486uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 BW-723C86 Adrenergic, Norepinephrine Transporter 78% 3.6257uM 3.5957uM View
Cytochrom P450-2D6 monooxygenase CYCLIZINE CYP450-2D6 Inhibition 78% 6.2175uM NoneNone View
epidermal growth factor receptor THIORIDAZINE Protein Tyrosine Kinase, EGF Receptor 78% 2.947uM NoneNone View
mitogen activated protein kinase 14 ZAFIRLUKAST Protein Serine/Threonine Kinase, p38alpha 78% .353uM NoneNone View
mitogen-activated protein kinase 14 ZAFIRLUKAST Protein Serine/Threonine Kinase, p38alpha 78% .353uM NoneNone View
cholinergic receptor, muscarinic 3 MONTELUKAST Muscarinic M3 78% 6.626uM 1.404uM View
cannabinoid receptor 1 (brain) FLUNARIZINE Cannabinoid CB1 78% 3.028uM 2.391uM View
calcium channel, voltage-dependent, gamma subunit 8 DIMENHYDRINATE Calcium Channel Type L, Phenylalkylamine 78% 3.344uM 3.251uM View
calcium channel, voltage-dependent, gamma subunit 7 DIMENHYDRINATE Calcium Channel Type L, Phenylalkylamine 78% 3.344uM 3.251uM View
calcium channel, voltage-dependent, gamma subunit 6 DIMENHYDRINATE Calcium Channel Type L, Phenylalkylamine 78% 3.344uM 3.251uM View
calcium channel, voltage-dependent, gamma subunit 5 DIMENHYDRINATE Calcium Channel Type L, Phenylalkylamine 78% 3.344uM 3.251uM View
calcium channel, voltage-dependent, gamma subunit 4 DIMENHYDRINATE Calcium Channel Type L, Phenylalkylamine 78% 3.344uM 3.251uM View
calcium channel, voltage-dependent, gamma subunit 3 DIMENHYDRINATE Calcium Channel Type L, Phenylalkylamine 78% 3.344uM 3.251uM View
calcium channel, voltage-dependent, gamma subunit 2 DIMENHYDRINATE Calcium Channel Type L, Phenylalkylamine 78% 3.344uM 3.251uM View
calcium channel, voltage-dependent, gamma subunit 1 DIMENHYDRINATE Calcium Channel Type L, Phenylalkylamine 78% 3.344uM 3.251uM View
sodium channel, voltage-gated, type III, beta PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide PROMAZINE Sodium Channel, Site 2 77% 2.573uM 2.347uM View
5-hydroxytryptamine (serotonin) receptor 2C TERCONAZOLE Serotonin 5-HT2C 77% 6.961uM 3.646uM View
adrenergic receptor, alpha 1d (Non-specific probe) TERCONAZOLE Adrenergic alpha1D 77% 14.385uM 7.07uM View
cholinergic receptor, muscarinic 2 PROCHLORPERAZINE Muscarinic M2 77% 3.112uM 1.107uM View
A3 adenosine receptor TROGLITAZONE Adenosine A3 77% 5.208uM 2.943uM View
adrenergic receptor, alpha 1d (Non-specific probe) ECONAZOLE Adrenergic alpha1D 77% 8.897uM 4.373uM View
calcium channel, voltage-dependent, gamma subunit 8 SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, gamma subunit 7 SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, gamma subunit 6 SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, gamma subunit 5 SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, gamma subunit 4 SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
Protein-tyrosine kinase, Fyn BETA-NAPHTHOFLAVONE Protein Tyrosine Kinase, Fyn 77% 2.5149uM NoneNone View
epidermal growth factor receptor PERHEXILINE Protein Tyrosine Kinase, EGF Receptor 77% 1.4852uM NoneNone View
Cytochrom P450-2C19 monooxygenase BUPROPION CYP450-2C19 Inhibition 77% 1.9983uM NoneNone View
5-hydroxytryptamine receptor 6 PROPAFENONE Serotonin 5-HT6 77% 1.863uM .865uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 AMBROXOL Serotonin Transporter 77% 3.391uM 1.802uM View
Protein-tyrosine kinase, Fyn TERFENADINE Protein Tyrosine Kinase, Fyn 77% 6.123uM NoneNone View
mu-opioid receptor MOR DOMPERIDONE Opiate mu 77% 4.218uM 1.712uM View
histamine receptor H 2 IMATINIB Histamine H2 77% 1.963uM 1.93uM View
dopamine receptor D3 CYCLIZINE Dopamine D3 77% 2.992uM 1.016uM View
Cytochrom P450-2D6 monooxygenase LOPERAMIDE CYP450-2D6 Inhibition 77% 2uM NoneNone View
Cytochrom P450-2C19 monooxygenase ETHYLESTRENOL CYP450-2C19 Inhibition 77% 1.2907uM NoneNone View
Cytochrom P450-2C19 monooxygenase RAPAMYCIN CYP450-2C19 Inhibition 77% 4uM NoneNone View
Cytochrom P450-2C19 monooxygenase RESVERATROL CYP450-2C19 Inhibition 77% 3uM NoneNone View
A3 adenosine receptor HYDROXYPROGESTERONE Adenosine A3 77% 4.73uM 2.674uM View
5-hydroxytryptamine (serotonin) receptor 2A DIPHENIDOL Serotonin 5-HT2A 77% 2.586uM .739uM View
estrogen receptor 1 ETHYLESTRENOL Estrogen ERalpha 77% 1.121uM .32uM View
estrogen receptor 1 ETHYLESTRENOL Estrogen ERalpha 77% 1.121uM .32uM View
adrenergic receptor, alpha 2a MOXONIDINE Imidazoline I2, Central 77% 1.4764uM .9843uM View
adrenergic receptor, alpha 2c (Non-specific probe) MOXONIDINE Imidazoline I2, Central 77% 1.4764uM .9843uM View
Protein-tyrosine kinase, Fyn METHYLDOPA Protein Tyrosine Kinase, Fyn 77% 5.176uM NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, gamma subunit 7 LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, gamma subunit 6 LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, gamma subunit 5 LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, gamma subunit 4 LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, gamma subunit 3 LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, gamma subunit 2 LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, gamma subunit 1 LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, beta 4 subunit LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, beta 3 subunit LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, beta 2 subunit LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, alpha 1F subunit LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, beta 1 subunit LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 LISURIDE Calcium Channel Type L, Benzothiazepine 77% 3.522uM 3.131uM View
epidermal growth factor receptor TERFENADINE Protein Tyrosine Kinase, EGF Receptor 76% 3.566uM NoneNone View
epidermal growth factor receptor ZAFIRLUKAST Protein Tyrosine Kinase, EGF Receptor 76% 5.751uM NoneNone View
angiotensin 1 converting enzyme 1 IODOQUINOL Protease, Angiotensin Converting Enzyme 76% .906uM NoneNone View
angiotensin I converting enzyme (peptidyl-dipeptidase A) 1 IODOQUINOL Protease, Angiotensin Converting Enzyme 76% .906uM NoneNone View
nitric oxide synthase 3 (endothelial cell) CHLORZOXAZONE Nitric Oxide Synthase, Constitutive (cNOS) 76% 2.794uM NoneNone View
nitric oxide synthase 3, endothelial cell CHLORZOXAZONE Nitric Oxide Synthase, Constitutive (cNOS) 76% 2.794uM NoneNone View
cholinergic receptor, muscarinic 4 CINNARIZINE Muscarinic M4 76% 3.66uM .51uM View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) ALPHA-ERGOCRYPTINE CYP450-2C9 Inhibition 76% 6uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 ALPHA-ERGOCRYPTINE CYP450-2C9 Inhibition 76% 6uM NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) RWJ-68354 CYP450-2C9 Inhibition 76% 1uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 RWJ-68354 CYP450-2C9 Inhibition 76% 1uM NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) PHENYLHYDRAZINE CYP450-2C9 Inhibition 76% 6uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 PHENYLHYDRAZINE CYP450-2C9 Inhibition 76% 6uM NoneNone View
Cytochrom P450-2C19 monooxygenase NOSCAPINE CYP450-2C19 Inhibition 76% .4003uM NoneNone View
adrenergic receptor, alpha 2b BERBERINE CHLORIDE Adrenergic alpha2C 76% 2.837uM .412uM View
adrenergic receptor, alpha 2c (Non-specific probe) BERBERINE CHLORIDE Adrenergic alpha2C 76% 2.837uM .412uM View
phosphodiesterase 3B MILRINONE Phosphodiesterase PDE3 76% .9585uM NoneNone View
phosphodiesterase 3A MILRINONE Phosphodiesterase PDE3 76% .9585uM NoneNone View
melanocortin 5 receptor DIGITONIN Melanocortin MC5 76% 3.88uM 3.639uM View
sodium channel, voltage-gated, type IV, beta MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel associated protein 1 MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel associated protein 2 MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type III, beta MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type I, alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type IX, alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type VII, alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
amiloride-sensitive cation channel 5, intestinal MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type III, beta MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type XI, alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type I, beta MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type 10, alpha polypeptide MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type IV, alpha polypeptide MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type V, alpha polypeptide MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type II, beta MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, nonvoltage-gated 1 alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, nonvoltage-gated 1 gamma MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, nonvoltage-gated 1 beta MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type XI, alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, nonvoltage-gated 1, gamma MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, nonvoltage-gated 1, delta MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, nonvoltage-gated 1 alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type X, alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type IX, alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage gated, type VIII, alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type VII, alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type IV, beta MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type IV, alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type III, alpha MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
sodium channel, voltage-gated, type II, beta MAPROTILINE Sodium Channel, Site 2 76% 2.572uM 2.346uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 CLEMASTINE Dopamine Transporter 89% .678uM .538uM View
adrenergic receptor, alpha 1d (Non-specific probe) CLEMASTINE Adrenergic alpha1D 89% .032uM .015uM View
5-hydroxytryptamine (serotonin) receptor 1B CLEMASTINE Serotonin 5-HT1B 89% .359uM .22uM View
calcium channel, voltage-dependent, gamma subunit 4 CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, gamma subunit 3 CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, gamma subunit 2 CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, gamma subunit 1 CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, beta 4 subunit CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, beta 3 subunit CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, beta 2 subunit CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, alpha 1F subunit CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, beta 1 subunit CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit CLEMASTINE Calcium Channel Type L, Phenylalkylamine 89% .508uM .493uM View
adrenergic receptor, alpha 2b DOMPERIDONE Adrenergic alpha2C 89% 1.011uM .147uM View
adrenergic receptor, alpha 2c (Non-specific probe) DOMPERIDONE Adrenergic alpha2C 89% 1.011uM .147uM View
cholinergic receptor, muscarinic 2 PENTAMIDINE Muscarinic M2 89% 1.425uM .507uM View
adrenergic receptor, alpha 2b EPINEPHRINE Adrenergic alpha2B 89% .869uM .397uM View
adrenergic receptor, alpha 2a METOCLOPRAMIDE Imidazoline I2, Central 89% .708uM .472uM View
adrenergic receptor, alpha 2c (Non-specific probe) METOCLOPRAMIDE Imidazoline I2, Central 89% .708uM .472uM View
calcium channel, voltage-dependent, gamma subunit 8 MICONAZOLE Calcium Channel Type L, Phenylalkylamine 89% 3.788uM 3.683uM View
calcium channel, voltage-dependent, gamma subunit 7 MICONAZOLE Calcium Channel Type L, Phenylalkylamine 89% 3.788uM 3.683uM View