Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
calcium channel, voltage-dependent, gamma subunit 5 DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 DIPHENIDOL Calcium Channel Type L, Benzothiazepine 66% NoneNone NoneNone View
epidermal growth factor receptor 3,3',4',5-TETRACHLOROSALICYLANILIDE Protein Tyrosine Kinase, EGF Receptor 66% NoneNone NoneNone View
cholinergic receptor, muscarinic 4 BITHIONOL Muscarinic M4 66% NoneNone NoneNone View
epidermal growth factor receptor GRAMICIDIN Protein Tyrosine Kinase, EGF Receptor 66% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 alpha BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, nonvoltage-gated 1 gamma BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, nonvoltage-gated 1 beta BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type XI, alpha BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, nonvoltage-gated 1, gamma BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, nonvoltage-gated 1, delta BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, nonvoltage-gated 1 alpha BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type X, alpha BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type IX, alpha BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage gated, type VIII, alpha BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type VII, alpha BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type IV, beta BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type IV, alpha BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type III, alpha BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type II, beta BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type II, alpha 2 BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type I, beta BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
sodium channel, voltage-gated, type I, alpha BROMOCRIPTINE Sodium Channel, Site 2 78% 6.692uM 6.105uM View
Sigma-2 Receptor EPERISONE Sigma2 78% 1.064uM .655uM View
calcium channel, voltage-dependent, gamma subunit 8 CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, gamma subunit 7 CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, gamma subunit 6 CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, gamma subunit 5 CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, gamma subunit 4 CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, gamma subunit 3 CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, gamma subunit 2 CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, gamma subunit 1 CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, beta 4 subunit CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, beta 3 subunit CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, beta 2 subunit CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, alpha 1F subunit CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, beta 1 subunit CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 CITALOPRAM Calcium Channel Type L, Phenylalkylamine 78% 1.025uM .996uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 CITALOPRAM Adrenergic, Norepinephrine Transporter 78% 2.196uM 2.178uM View
thromboxane A synthase 1 INDINAVIR Thromboxane Synthetase 78% 1.851uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) INDINAVIR Thromboxane Synthetase 78% 1.851uM NoneNone View
adrenergic receptor, beta 2 MONTELUKAST Adrenergic beta2 78% 3.488uM 2.398uM View
5-hydroxytryptamine (serotonin) receptor 2B 1-(2-CHLOROBENZOYL)-4-(PHENYLMETHYL)-PIPERIDINE Serotonin 5-HT2B 78% 1.508uM .96uM View
Sigma-2 Receptor LOPERAMIDE Sigma2 78% 1.379uM .848uM View
opioid receptor, sigma 1 PROPRANOLOL Sigma1 78% 2.87uM 1.206uM View
sodium channel, voltage-gated, type II, alpha 2 CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type I, beta CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type I, alpha CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type IV, beta CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel associated protein 1 CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel associated protein 2 CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type III, beta CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type I, alpha CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type IX, alpha CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type VII, alpha CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
amiloride-sensitive cation channel 5, intestinal CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type III, beta CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type XI, alpha CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type I, beta CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type 10, alpha polypeptide CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type IV, alpha polypeptide CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type V, alpha polypeptide CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type II, beta CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, nonvoltage-gated 1 alpha CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, nonvoltage-gated 1 gamma CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, nonvoltage-gated 1 beta CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, voltage-gated, type XI, alpha CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
sodium channel, nonvoltage-gated 1, gamma CITALOPRAM Sodium Channel, Site 2 77% 2.641uM 2.409uM View
5-hydroxytryptamine (serotonin) receptor 3a MIANSERIN Serotonin 5-HT3 77% 2.746uM .617uM View
5-hydroxytryptamine (serotonin) receptor 3b MIANSERIN Serotonin 5-HT3 77% 2.746uM .617uM View
adrenergic receptor, beta 2 LOPERAMIDE Adrenergic beta2 77% 3.005uM 2.066uM View
5-hydroxytryptamine (serotonin) receptor 2B 4-(PHENYLMETHYL)-1-[2-(TRIFLUOROMETHYL)BENZOYL]-PIPERIDINE Serotonin 5-HT2B 77% 1.549uM .986uM View
calcium channel, voltage-dependent, gamma subunit 3 SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, gamma subunit 2 SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, gamma subunit 1 SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, beta 4 subunit SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
sodium channel associated protein 2 PUROMYCIN Sodium Channel, Site 2 12% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, beta 2 subunit SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, alpha 1F subunit SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, beta 1 subunit SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 SULCONAZOLE Calcium Channel Type L, Dihydropyridine 77% 2.427uM 1.56uM View
phosphodiesterase 3B DANAZOL Phosphodiesterase PDE3 77% 2.535uM NoneNone View
phosphodiesterase 3A DANAZOL Phosphodiesterase PDE3 77% 2.535uM NoneNone View
Protein-tyrosine kinase, Fyn SULCONAZOLE Protein Tyrosine Kinase, Fyn 77% 3.704uM NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 DIETHYLSTILBESTROL Calcium Channel Type L, Phenylalkylamine 77% 3.761uM 3.65uM View
calcium channel, voltage-dependent, gamma subunit 7 DIETHYLSTILBESTROL Calcium Channel Type L, Phenylalkylamine 77% 3.761uM 3.65uM View
calcium channel, voltage-dependent, gamma subunit 6 DIETHYLSTILBESTROL Calcium Channel Type L, Phenylalkylamine 77% 3.761uM 3.65uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit OXICONAZOLE Calcium Channel Type L, Phenylalkylamine 76% 2.7269uM 2.6512uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit OXICONAZOLE Calcium Channel Type L, Phenylalkylamine 76% 2.7269uM 2.6512uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit OXICONAZOLE Calcium Channel Type L, Phenylalkylamine 76% 2.7269uM 2.6512uM View
calcium channel, voltage-dependent, beta 1 subunit OXICONAZOLE Calcium Channel Type L, Phenylalkylamine 76% 2.7269uM 2.6512uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit OXICONAZOLE Calcium Channel Type L, Phenylalkylamine 76% 2.7269uM 2.6512uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit OXICONAZOLE Calcium Channel Type L, Phenylalkylamine 76% 2.7269uM 2.6512uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 OXICONAZOLE Calcium Channel Type L, Phenylalkylamine 76% 2.7269uM 2.6512uM View
cholinergic receptor, muscarinic 1 OXICONAZOLE Muscarinic M1 76% 4.7364uM 1.1407uM View
Sigma-2 Receptor PRAMOXINE Sigma2 76% 1.029uM .633uM View
thromboxane A synthase 1 AMPRENAVIR Thromboxane Synthetase 76% 6.727uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) AMPRENAVIR Thromboxane Synthetase 76% 6.727uM NoneNone View
melanocortin 4 receptor CETYLPYRIDINIUM BROMIDE Melanocortin MC4 76% 5.081uM 4.886uM View
dopamine receptor D1A RALOXIFENE Dopamine D1 76% 3.864uM 1.932uM View
ATP-binding cassette, sub-family C (CFTR/MRP), member 8 NATEGLINIDE Potassium Channel [KATP] 76% 1.667uM .189uM View
ATP-binding cassette, sub-family C (CFTR/MRP), member 9 NATEGLINIDE Potassium Channel [KATP] 76% 1.667uM .189uM View
ATP-binding cassette, sub-family C (CFTR/MRP), member 8 NATEGLINIDE Potassium Channel [KATP] 76% 1.667uM .189uM View
lymphocyte protein tyrosine kinase (mapped) TRIBROMSALAN Protein Tyrosine Kinase, Lck 76% 5.015uM NoneNone View
tachykinin receptor 2 CLOMIPHENE Tachykinin NK2 76% 4.525uM 1.508uM View
adrenergic receptor, beta 1 ATENOLOL Adrenergic beta1 76% 1.313uM .758uM View
calcium channel, voltage-dependent, gamma subunit 1 PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, beta 4 subunit PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, beta 3 subunit PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, beta 2 subunit PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
sodium channel, voltage-gated, type III, beta PUROMYCIN Sodium Channel, Site 2 12% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, beta 1 subunit PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 PERGOLIDE Calcium Channel Type L, Phenylalkylamine 76% .913uM .887uM View
5-hydroxytryptamine (serotonin) receptor 1B CYPROHEPTADINE Serotonin 5-HT1B 76% 2.778uM 1.263uM View
cysteinyl leukotriene receptor 1 GW-1929 Leukotriene D4 76% 10.91uM 5.455uM View
cysteinyl leukotriene receptor 1 GW-1929 Leukotriene D4 76% 10.91uM 5.455uM View
5-hydroxytryptamine (serotonin) receptor 2C METOCLOPRAMIDE Serotonin 5-HT2C 76% 2.383uM 1.248uM View
histamine receptor H 2 ECONAZOLE Histamine H2 76% 1.592uM 1.565uM View
melanocortin 3 receptor MICONAZOLE Melanocortin MC3 76% 18.485uM 16.132uM View
melanocortin 3 receptor MICONAZOLE Melanocortin MC3 76% 18.485uM 16.132uM View
cholinergic receptor, muscarinic 4 CIGLITAZONE Muscarinic M4 76% 16.224uM 2.263uM View
cysteinyl leukotriene receptor 1 DIETHYLSTILBESTROL Leukotriene D4 76% 17.745uM 8.872uM View
cysteinyl leukotriene receptor 1 DIETHYLSTILBESTROL Leukotriene D4 76% 17.745uM 8.872uM View
androgen receptor ESTRONE Testosterone 76% 11.617uM 7.745uM View
Cytochrom P450-2D6 monooxygenase AJMALINE CYP450-2D6 Inhibition 76% 1uM NoneNone View
Cytochrom P450-1A2 monooxygenase 3-METHYLCHOLANTHRENE CYP450-1A2 Inhibition 76% .3uM NoneNone View
Protein-tyrosine kinase, Fyn PACLITAXEL Protein Tyrosine Kinase, Fyn 76% 23.906uM NoneNone View
lymphocyte protein tyrosine kinase (mapped) TANNIC ACID Protein Tyrosine Kinase, Lck 76% .079uM NoneNone View
leukotriene C4 synthase TANNIC ACID Leukotriene C4 Synthetase 76% 2.715uM NoneNone View
leukotriene C4 synthase TANNIC ACID Leukotriene C4 Synthetase 76% 2.715uM NoneNone View
dopamine receptor D3 U-78517F Dopamine D3 76% 5.196uM 1.765uM View
calcium channel, voltage-dependent, gamma subunit 8 CLOTRIMAZOLE Calcium Channel Type L, Phenylalkylamine 76% 2.478uM 2.41uM View
calcium channel, voltage-dependent, gamma subunit 7 CLOTRIMAZOLE Calcium Channel Type L, Phenylalkylamine 76% 2.478uM 2.41uM View
calcium channel, voltage-dependent, gamma subunit 6 CLOMIPHENE Calcium Channel Type L, Dihydropyridine 75% 1.62uM 1.041uM View
calcium channel, voltage-dependent, gamma subunit 5 CLOMIPHENE Calcium Channel Type L, Dihydropyridine 75% 1.62uM 1.041uM View
calcium channel, voltage-dependent, gamma subunit 4 CLOMIPHENE Calcium Channel Type L, Dihydropyridine 75% 1.62uM 1.041uM View
calcium channel, voltage-dependent, gamma subunit 3 CLOMIPHENE Calcium Channel Type L, Dihydropyridine 75% 1.62uM 1.041uM View
calcium channel, voltage-dependent, gamma subunit 2 CLOMIPHENE Calcium Channel Type L, Dihydropyridine 75% 1.62uM 1.041uM View
calcium channel, voltage-dependent, gamma subunit 1 CLOMIPHENE Calcium Channel Type L, Dihydropyridine 75% 1.62uM 1.041uM View
calcium channel, voltage-dependent, beta 4 subunit CLOMIPHENE Calcium Channel Type L, Dihydropyridine 75% 1.62uM 1.041uM View
calcium channel, voltage-dependent, beta 3 subunit CLOMIPHENE Calcium Channel Type L, Dihydropyridine 75% 1.62uM 1.041uM View
adrenergic receptor, alpha 2b GUANFACINE Adrenergic alpha2C 75% 6.447uM .937uM View
adrenergic receptor, alpha 2c (Non-specific probe) GUANFACINE Adrenergic alpha2C 75% 6.447uM .937uM View
adrenergic receptor, alpha 1a VERAPAMIL Adrenergic alpha1A 75% 2.092uM .847uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 2-ACETYLAMINOFLUORENE Adrenergic, Norepinephrine Transporter 75% 8.595uM 8.524uM View
A3 adenosine receptor MITOTANE Adenosine A3 75% 7.445uM 4.208uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 N,N'-DIPHENYL-P-PHENYLENEDIAMINE Adrenergic, Norepinephrine Transporter 75% .786uM .78uM View
5-hydroxytryptamine receptor 6 PROPRANOLOL Serotonin 5-HT6 75% 3.065uM 1.423uM View
5-hydroxytryptamine (serotonin) receptor 2C MITOXANTRONE Serotonin 5-HT2C 75% 3.5619uM 1.8657uM View
adrenergic receptor, alpha 2b IRINOTECAN Adrenergic alpha2C 75% 3.171uM .461uM View
adrenergic receptor, alpha 2c (Non-specific probe) IRINOTECAN Adrenergic alpha2C 75% 3.171uM .461uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 QUINACRINE Adrenergic, Norepinephrine Transporter 75% 2.896uM 2.872uM View
adenosine A2a receptor IMIQUIMOD Adenosine A2A 75% 5.32uM 2.987uM View
5-hydroxytryptamine (serotonin) receptor 1A KETOTIFEN Serotonin 5-HT1A 75% 2.537uM 1.45uM View
adrenergic receptor, alpha 1d (Non-specific probe) KETOTIFEN Adrenergic alpha1D 75% 3.727uM 1.832uM View
Sigma-2 Receptor SERTRALINE Sigma2 75% 2.119uM 1.304uM View
calcium channel, voltage-dependent, gamma subunit 8 NORTRIPTYLINE Calcium Channel Type L, Benzothiazepine 75% 2.803uM 2.492uM View
calcium channel, voltage-dependent, gamma subunit 7 NORTRIPTYLINE Calcium Channel Type L, Benzothiazepine 75% 2.803uM 2.492uM View
calcium channel, voltage-dependent, gamma subunit 6 NORTRIPTYLINE Calcium Channel Type L, Benzothiazepine 75% 2.803uM 2.492uM View
calcium channel, voltage-dependent, gamma subunit 5 NORTRIPTYLINE Calcium Channel Type L, Benzothiazepine 75% 2.803uM 2.492uM View