Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
calcium channel, voltage-dependent, L type, alpha 1E subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, gamma subunit 8 FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, gamma subunit 7 FLUOXETINE Calcium Channel Type L, Phenylalkylamine 94% 1.126uM 1.095uM View
calcium channel, voltage-dependent, alpha 1F subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, beta 1 subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 DESLORATADINE Calcium Channel Type L, Benzothiazepine 73% 5.791uM 5.148uM View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) RESVERATROL CYP450-2C9 Inhibition 73% 7uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 RESVERATROL CYP450-2C9 Inhibition 73% 7uM NoneNone View
calcium channel, voltage-dependent, beta 2 subunit MAPROTILINE Calcium Channel Type L, Phenylalkylamine 71% .446uM .434uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit MAPROTILINE Calcium Channel Type L, Phenylalkylamine 71% .446uM .434uM View
calcium channel, voltage-dependent, alpha 1F subunit MAPROTILINE Calcium Channel Type L, Phenylalkylamine 71% .446uM .434uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit MAPROTILINE Calcium Channel Type L, Phenylalkylamine 71% .446uM .434uM View
calcium channel, voltage-dependent, alpha 1F subunit DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 DOXEPIN Calcium Channel Type L, Benzothiazepine 69% NoneNone NoneNone View
adrenergic receptor, alpha 2b SULPIRIDE Adrenergic alpha2B 69% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, beta LABETALOL Sodium Channel, Site 2 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit NELFINAVIR Calcium Channel Type L, Phenylalkylamine 69% 18.38uM 17.862uM View
calcium channel, voltage-dependent, beta 3 subunit NELFINAVIR Calcium Channel Type L, Phenylalkylamine 69% 18.38uM 17.862uM View
calcium channel, voltage-dependent, beta 2 subunit NELFINAVIR Calcium Channel Type L, Phenylalkylamine 69% 18.38uM 17.862uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit NELFINAVIR Calcium Channel Type L, Phenylalkylamine 69% 18.38uM 17.862uM View
calcium channel, voltage-dependent, alpha 1F subunit NELFINAVIR Calcium Channel Type L, Phenylalkylamine 69% 18.38uM 17.862uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit NELFINAVIR Calcium Channel Type L, Phenylalkylamine 69% 18.38uM 17.862uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit NELFINAVIR Calcium Channel Type L, Phenylalkylamine 69% 18.38uM 17.862uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit NELFINAVIR Calcium Channel Type L, Phenylalkylamine 69% 18.38uM 17.862uM View
calcium channel, voltage-dependent, beta 1 subunit NELFINAVIR Calcium Channel Type L, Phenylalkylamine 69% 18.38uM 17.862uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit NELFINAVIR Calcium Channel Type L, Phenylalkylamine 69% 18.38uM 17.862uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit NELFINAVIR Calcium Channel Type L, Phenylalkylamine 69% 18.38uM 17.862uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 NELFINAVIR Calcium Channel Type L, Phenylalkylamine 69% 18.38uM 17.862uM View
histamine receptor H 2 NIZATIDINE Histamine H2 69% NoneNone NoneNone View
adrenergic receptor, alpha 2b CYCLIZINE Adrenergic alpha2C 69% NoneNone NoneNone View
adrenergic receptor, alpha 2c (Non-specific probe) CYCLIZINE Adrenergic alpha2C 69% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 ETHYNODIOL DIACETATE Adrenergic, Norepinephrine Transporter 69% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 FENOFIBRATE Dopamine Transporter 69% 8.633uM 6.859uM View
calcium channel, voltage-dependent, gamma subunit 7 SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 6 SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 5 SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 4 SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 3 SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 2 SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 1 SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 4 subunit SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 3 subunit SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 2 subunit SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1S subunit SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha 1F subunit SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) DACTINOMYCIN Protein Tyrosine Kinase, HER2 Receptor 66% NoneNone NoneNone View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) DACTINOMYCIN Protein Tyrosine Kinase, HER2 Receptor 66% NoneNone NoneNone View
mitogen activated protein kinase 3 GRAMICIDIN Protein Serine/Threonine Kinase, ERK1 66% NoneNone NoneNone View
mitogen-activated protein kinase 3 GRAMICIDIN Protein Serine/Threonine Kinase, ERK1 66% NoneNone NoneNone View
dopamine receptor D4 PROMAZINE Dopamine D4.2 66% NoneNone NoneNone View
adrenergic receptor, alpha 1b TERCONAZOLE Adrenergic alpha1B 66% 14.299uM 7.915uM View
cholinergic receptor, muscarinic 2 PRIMAQUINE Muscarinic M2 65% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 TERCONAZOLE Serotonin Transporter 66% 11.456uM 6.086uM View
adrenergic receptor, alpha 1d (Non-specific probe) TERFENADINE Adrenergic alpha1D 66% NoneNone NoneNone View
mitogen activated protein kinase 3 NELFINAVIR Protein Serine/Threonine Kinase, ERK1 66% 22.503uM NoneNone View
mitogen-activated protein kinase 3 NELFINAVIR Protein Serine/Threonine Kinase, ERK1 66% 22.503uM NoneNone View
acetylcholinesterase (YT blood group) TERCONAZOLE Acetylcholinesterase 66% 21.573uM NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase TERCONAZOLE Acetylcholinesterase 66% 21.573uM NoneNone View
acetylcholinesterase TERCONAZOLE Acetylcholinesterase 66% 21.573uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 1B PENTAMIDINE Serotonin 5-HT1B 66% NoneNone NoneNone View
epidermal growth factor receptor PROCHLORPERAZINE Protein Tyrosine Kinase, EGF Receptor 66% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 S-(-)-PROPRANOLOL Adrenergic, Norepinephrine Transporter 66% NoneNone NoneNone View
melanocortin 4 receptor GUANABENZ Melanocortin MC4 66% NoneNone NoneNone View
ATPase, Na+/K+ transporting, alpha 4 polypeptide MICONAZOLE ATPase, Na+/K+ 66% 19.279uM NoneNone View
ATPase, Na+/K+ transporting, alpha 3 polypeptide MICONAZOLE ATPase, Na+/K+ 66% 19.279uM NoneNone View
ATPase, Na+/K+ transporting, alpha 2 polypeptide MICONAZOLE ATPase, Na+/K+ 66% 19.279uM NoneNone View
ATPase, Na+/K+ transporting, alpha 1 polypeptide MICONAZOLE ATPase, Na+/K+ 66% 19.279uM NoneNone View
calcium channel, voltage-dependent, L type, alpha 1D subunit EMETINE Calcium Channel Type L, Phenylalkylamine 65% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit EMETINE Calcium Channel Type L, Phenylalkylamine 65% NoneNone NoneNone View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit EMETINE Calcium Channel Type L, Phenylalkylamine 65% NoneNone NoneNone View
calcium channel, voltage-dependent, beta 1 subunit EMETINE Calcium Channel Type L, Phenylalkylamine 65% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit EMETINE Calcium Channel Type L, Phenylalkylamine 65% NoneNone NoneNone View
calcium channel, voltage-dependent, N type, alpha 1B subunit EMETINE Calcium Channel Type L, Phenylalkylamine 65% NoneNone NoneNone View
calcium channel, voltage-dependent, alpha2/delta subunit 1 EMETINE Calcium Channel Type L, Phenylalkylamine 65% NoneNone NoneNone View
opioid receptor, sigma 1 DIPHENHYDRAMINE Sigma1 65% NoneNone NoneNone View
histamine receptor H 2 DIPHENHYDRAMINE Histamine H2 65% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 TROGLITAZONE Adrenergic, Norepinephrine Transporter 65% NoneNone NoneNone View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 RESERPINE Adrenergic, Norepinephrine Transporter 65% NoneNone NoneNone View
mu-opioid receptor MOR CADMIUM CHLORIDE Opiate mu 65% NoneNone NoneNone View
lymphocyte protein tyrosine kinase (mapped) CADMIUM CHLORIDE Protein Tyrosine Kinase, Lck 65% NoneNone NoneNone View
interleukin 8 receptor, beta CETYLPYRIDINIUM BROMIDE Chemokine CXCR2 (IL-8B) 65% NoneNone NoneNone View
sodium channel, voltage-gated, type II, beta SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 alpha SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 gamma SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 beta SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, voltage-gated, type XI, alpha SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, gamma SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, delta SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 alpha SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, voltage-gated, type X, alpha SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, voltage-gated, type IX, alpha SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, voltage gated, type VIII, alpha SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, voltage-gated, type VII, alpha SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, voltage-gated, type V, alpha (long QT syndrome 3) SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, beta SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, alpha SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
sodium channel, voltage-gated, type III, alpha SIBUTRAMINE Sodium Channel, Site 2 65% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1C subunit MAPROTILINE Calcium Channel Type L, Phenylalkylamine 71% .446uM .434uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit MAPROTILINE Calcium Channel Type L, Phenylalkylamine 71% .446uM .434uM View
calcium channel, voltage-dependent, beta 1 subunit MAPROTILINE Calcium Channel Type L, Phenylalkylamine 71% .446uM .434uM View
sodium channel, voltage-gated, type I, alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
calcium channel, voltage-dependent, L type, alpha 1E subunit MAPROTILINE Calcium Channel Type L, Phenylalkylamine 71% .446uM .434uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit MAPROTILINE Calcium Channel Type L, Phenylalkylamine 71% .446uM .434uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 MAPROTILINE Calcium Channel Type L, Phenylalkylamine 71% .446uM .434uM View
lymphocyte protein tyrosine kinase (mapped) ERGOTAMINE Protein Tyrosine Kinase, Lck 71% 6.499uM NoneNone View
adrenergic receptor, beta 2 ERGOTAMINE Adrenergic beta2 71% 2.761uM 1.898uM View
sodium channel, voltage-gated, type IV, beta PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel associated protein 1 PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel associated protein 2 PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type III, beta PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type I, alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type IX, alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type VII, alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
amiloride-sensitive cation channel 5, intestinal PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type III, beta PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type XI, alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type I, beta PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type 10, alpha polypeptide PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type IV, alpha polypeptide PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type V, alpha polypeptide PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type II, beta PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, nonvoltage-gated 1 alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, nonvoltage-gated 1 gamma PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, nonvoltage-gated 1 beta PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, voltage-gated, type XI, alpha PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
sodium channel, nonvoltage-gated 1, gamma PYRILAMINE Sodium Channel, Site 2 71% 5.283uM 4.819uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 TRIHEXYPHENIDYL Calcium Channel Type L, Benzothiazepine 70% 4.81uM 4.275uM View
calcium channel, voltage-dependent, beta 3 subunit QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, beta 2 subunit QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, alpha 1F subunit QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, beta 1 subunit QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 QUINACRINE Calcium Channel Type L, Benzothiazepine 70% 1.076uM .956uM View
histamine receptor H 2 NORTRIPTYLINE Histamine H2 70% 2.334uM 2.295uM View
5-hydroxytryptamine (serotonin) receptor 1B NORTRIPTYLINE Serotonin 5-HT1B 70% 3.199uM 1.454uM View
adrenergic receptor, alpha 2a NORTRIPTYLINE Imidazoline I2, Central 70% 3.858uM 2.572uM View
adrenergic receptor, alpha 2c (Non-specific probe) NORTRIPTYLINE Imidazoline I2, Central 70% 3.858uM 2.572uM View
A3 adenosine receptor STANOZOLOL Adenosine A3 70% 8.325uM 4.705uM View
adrenergic receptor, alpha 2b RALOXIFENE Adrenergic alpha2B 70% 3.698uM 1.688uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 SIBUTRAMINE Adrenergic, Norepinephrine Transporter 70% 5.665uM 5.619uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 SULCONAZOLE Calcium Channel Type L, Phenylalkylamine 69% NoneNone NoneNone View
adrenergic receptor, beta 3 SULCONAZOLE Adrenergic beta3 69% NoneNone NoneNone View
mu-opioid receptor MOR DANAZOL Opiate mu 69% 14.079uM 5.715uM View
Protein-tyrosine kinase, Fyn BETA-ESTRADIOL 3-BENZOATE Protein Tyrosine Kinase, Fyn 69% 22.994uM NoneNone View
sodium channel associated protein 2 AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type III, beta AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type IX, alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type VII, alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
amiloride-sensitive cation channel 5, intestinal AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type III, beta AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type VIII, alpha polypeptide AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type XI, alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type I, beta AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type 10, alpha polypeptide AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, alpha polypeptide AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type V, alpha polypeptide AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type II, beta AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 gamma AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1 beta AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, voltage-gated, type XI, alpha AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
sodium channel, nonvoltage-gated 1, gamma AMOXAPINE Sodium Channel, Site 2 69% NoneNone NoneNone View
monoamine oxidase A BETA-NAPHTHOFLAVONE Monoamine Oxidase MAOA 69% NoneNone NoneNone View
monoamine oxidase A BETA-NAPHTHOFLAVONE Monoamine Oxidase MAOA 69% NoneNone NoneNone View
opioid receptor, sigma 1 METHAPYRILENE Sigma1 69% NoneNone NoneNone View
5-hydroxytryptamine receptor 6 DIMENHYDRINATE Serotonin 5-HT6 69% NoneNone NoneNone View
cytochrome P450, family 3, subfamily a, polypeptide 13 MYCOPHENOLATE MOFETIL CYP450-3A4 Inhibition 69% NoneNone NoneNone View
Cytochrom P450-2C19 monooxygenase PROCHLORPERAZINE CYP450-2C19 Inhibition 69% NoneNone NoneNone View
Sigma-2 Receptor BUFLOMEDIL Sigma2 69% NoneNone NoneNone View
Cytochrom P450-1A2 monooxygenase 3,3',4',5-TETRACHLOROSALICYLANILIDE CYP450-1A2 Inhibition 69% NoneNone NoneNone View