Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
sodium channel, voltage-gated, type II, beta ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type II, alpha 2 ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type I, beta ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type I, alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type IV, beta ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel associated protein 1 ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel associated protein 2 ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type III, beta ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type I, alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type IX, alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
5-hydroxytryptamine (serotonin) receptor 2B N,N'-DIPHENYL-P-PHENYLENEDIAMINE Serotonin 5-HT2B 92% .142uM .09uM View
5-hydroxytryptamine (serotonin) receptor 2B PROPRANOLOL Serotonin 5-HT2B 92% .342uM .218uM View
glutamate receptor, ionotropic, N-methyl D-aspartate 2D KETAMINE Glutamate, NMDA, Phencyclidine 92% 1.01uM .684uM View
glutamate receptor, ionotropic, NMDA2C KETAMINE Glutamate, NMDA, Phencyclidine 92% 1.01uM .684uM View
glutamate receptor, ionotropic, N-methyl D-aspartate 2B KETAMINE Glutamate, NMDA, Phencyclidine 92% 1.01uM .684uM View
glutamate receptor, ionotropic, N-methyl D-aspartate 2A KETAMINE Glutamate, NMDA, Phencyclidine 92% 1.01uM .684uM View
N-methyl-D-aspartate receptor 1 (Grin1) gene, exons 1 through 6 and partial cds; alternatively spliced (Rn.) KETAMINE Glutamate, NMDA, Phencyclidine 92% 1.01uM .684uM View
glutamate receptor, ionotropic, N-methyl-D-aspartate 3B KETAMINE Glutamate, NMDA, Phencyclidine 92% 1.01uM .684uM View
adrenergic receptor, beta 3 BOPINDOLOL Adrenergic beta3 92% .458uM .344uM View
nuclear receptor subfamily 3, group C, member 1 CYPROTERONE ACETATE Glucocorticoid 92% .225uM .102uM View
calcium channel, voltage-dependent, gamma subunit 8 RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, gamma subunit 7 RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, gamma subunit 6 RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, gamma subunit 5 RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, gamma subunit 4 RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, gamma subunit 3 RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, gamma subunit 2 RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, gamma subunit 1 RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, beta 4 subunit RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, beta 3 subunit RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, beta 2 subunit RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, alpha 1F subunit RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, beta 1 subunit RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 RESERPINE Calcium Channel Type L, Dihydropyridine 92% .821uM .528uM View
adrenergic receptor, alpha 1d (Non-specific probe) OLANZAPINE Adrenergic alpha1D 92% .092uM .045uM View
dopamine receptor 2 OLANZAPINE Dopamine D2L 92% .118uM .039uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 OXICONAZOLE Adrenergic, Norepinephrine Transporter 92% 1.9103uM 1.8945uM View
calcium channel, voltage-dependent, gamma subunit 8 EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, gamma subunit 7 EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, gamma subunit 6 EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, gamma subunit 5 EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, gamma subunit 4 EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, gamma subunit 3 EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, gamma subunit 2 EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, gamma subunit 1 EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, beta 4 subunit EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, beta 3 subunit EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
sodium channel, voltage-gated, type III, beta ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type VIII, alpha polypeptide ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type XI, alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type I, beta ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type 10, alpha polypeptide ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type IV, alpha polypeptide ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type V, alpha polypeptide ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type II, beta ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, nonvoltage-gated 1 alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, nonvoltage-gated 1 gamma ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, nonvoltage-gated 1 beta ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type 2, alpha 1 polypeptide ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type XI, alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, nonvoltage-gated 1, gamma ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, nonvoltage-gated 1, delta ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, nonvoltage-gated 1, beta (Liddle syndrome) ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, nonvoltage-gated 1 alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type X, alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type IX, alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage gated, type VIII, alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
sodium channel, voltage-gated, type VII, alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 KETOCONAZOLE Serotonin Transporter 92% .531uM .282uM View
5-hydroxytryptamine (serotonin) receptor 2C DEXCHLORPHENIRAMINE Serotonin 5-HT2C 92% 2.322uM 1.217uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 DEXCHLORPHENIRAMINE Dopamine Transporter 92% .931uM .739uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 CIGLITAZONE Serotonin Transporter 92% 14.948uM 7.941uM View
dopamine receptor D1A ERGOCORNINE Dopamine D1 92% .294uM .147uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 SULCONAZOLE Dopamine Transporter 92% 1.726uM 1.371uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 DANAZOL Adrenergic, Norepinephrine Transporter 92% 5.698uM 5.651uM View
dopamine receptor D1A DIETHYLSTILBESTROL Dopamine D1 92% 7.763uM 3.882uM View
mu-opioid receptor MOR MIFEPRISTONE Opiate mu 92% 2.457uM .997uM View
adrenergic receptor, alpha 1d (Non-specific probe) EPINEPHRINE Adrenergic alpha1D 92% .449uM .221uM View
prostaglandin-endoperoxide synthase 2 4-OCTYLPHENOL Cyclooxygenase COX-2 92% 2.862uM NoneNone View
prostaglandin-endoperoxide synthase 2 (prostaglandin G/H synthase and cyclooxygenase) 4-OCTYLPHENOL Cyclooxygenase COX-2 92% 2.862uM NoneNone View
epidermal growth factor receptor PYROGALLOL Protein Tyrosine Kinase, EGF Receptor 92% 1.23uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 CELECOXIB Serotonin Transporter 92% 6.276uM 3.334uM View
phosphodiesterase 5A, cGMP-specific ALPHA-NAPHTHOFLAVONE Phosphodiesterase PDE5 92% 2.3034uM NoneNone View
phosphodiesterase 5A, cGMP-specific ALPHA-NAPHTHOFLAVONE Phosphodiesterase PDE5 92% 2.3034uM NoneNone View
thromboxane A synthase 1 CLOTRIMAZOLE Thromboxane Synthetase 92% .014uM NoneNone View
thromboxane A synthase 1 (platelet, cytochrome P450, family 5, subfamily A) CLOTRIMAZOLE Thromboxane Synthetase 92% .014uM NoneNone View
mitogen activated protein kinase 1 TRETINOIN Protein Serine/Threonine Kinase, ERK2 92% .576uM NoneNone View
mitogen-activated protein kinase 1 TRETINOIN Protein Serine/Threonine Kinase, ERK2 92% .576uM NoneNone View
cholinergic receptor, muscarinic 4 BETAMETHASONE PHOSPHATE Muscarinic M4 92% 11.924uM 1.663uM View
calcium channel, voltage-dependent, gamma subunit 8 TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, gamma subunit 7 TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, gamma subunit 6 TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, gamma subunit 5 TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, gamma subunit 4 TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, gamma subunit 3 TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, gamma subunit 2 TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, gamma subunit 1 TAMOXIFEN Calcium Channel Type L, Phenylalkylamine 92% 2.042uM 1.985uM View
calcium channel, voltage-dependent, beta 2 subunit EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, alpha 1F subunit EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, beta 1 subunit EBASTINE Calcium Channel Type L, Dihydropyridine 92% .1436uM .0923uM View
calcium channel, voltage-dependent, gamma subunit 1 DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, beta 4 subunit DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, beta 3 subunit DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, beta 2 subunit DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, alpha 1F subunit DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, beta 1 subunit DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, gamma subunit 8 DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, gamma subunit 7 DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, gamma subunit 6 DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, gamma subunit 5 DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
calcium channel, voltage-dependent, gamma subunit 4 DICYCLOMINE Calcium Channel Type L, Phenylalkylamine 92% .11uM .107uM View
prostaglandin-endoperoxide synthase 1 ASPIRIN Cyclooxygenase COX-1 92% 4.192uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) ASPIRIN Cyclooxygenase COX-1 92% 4.192uM NoneNone View
progesterone receptor FLURANDRENOLIDE Progesterone 92% .172uM .022uM View
progesterone receptor FLURANDRENOLIDE Progesterone 92% .172uM .022uM View
opioid receptor, sigma 1 TICLOPIDINE Sigma1 92% .426uM .179uM View
prostaglandin-endoperoxide synthase 1 FLURBIPROFEN Cyclooxygenase COX-1 92% .021uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) FLURBIPROFEN Cyclooxygenase COX-1 92% .021uM NoneNone View
adrenergic receptor, alpha 2a TICLOPIDINE Adrenergic alpha2A 92% .382uM .143uM View
prostaglandin-endoperoxide synthase 2 SULINDAC SULFIDE Cyclooxygenase COX-2 92% 1.537uM NoneNone View
prostaglandin-endoperoxide synthase 2 (prostaglandin G/H synthase and cyclooxygenase) SULINDAC SULFIDE Cyclooxygenase COX-2 92% 1.537uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 R-(+)-PROPRANOLOL Serotonin Transporter 92% .612uM .325uM View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 GENTIAN VIOLET Dopamine Transporter 92% 4.069uM 3.233uM View
dopamine receptor D1A MIANSERIN Dopamine D1 92% .543uM .271uM View
adrenergic receptor, alpha 2a MIANSERIN Imidazoline I2, Central 92% .124uM .083uM View
adrenergic receptor, alpha 2c (Non-specific probe) MIANSERIN Imidazoline I2, Central 92% .124uM .083uM View
tachykinin receptor 2 INDINAVIR Tachykinin NK2 92% 5.101uM 1.7uM View
dopamine receptor 2 LYSERGOL Dopamine D2L 92% .702uM .234uM View
adrenergic receptor, alpha 1b LOPERAMIDE Adrenergic alpha1B 92% .965uM .534uM View
histamine receptor H 1 LORATADINE Histamine H1, Central 92% .17uM .02uM View
adenosine A1 receptor RWJ-68354 Adenosine A1 92% .887uM .518uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 RWJ-68354 Adrenergic, Norepinephrine Transporter 92% 1.07uM 1.061uM View
5-hydroxytryptamine (serotonin) receptor 1A RISPERIDONE Serotonin 5-HT1A 92% .799uM .457uM View
dopamine receptor D1A RISPERIDONE Dopamine D1 92% .479uM .24uM View
sodium channel, voltage-gated, type VII, alpha ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
amiloride-sensitive cation channel 5, intestinal ITRACONAZOLE Sodium Channel, Site 2 92% 2.577uM 2.351uM View
angiotensin 1 converting enzyme 1 CAPTOPRIL Protease, Angiotensin Converting Enzyme 93% .13uM NoneNone View
angiotensin I converting enzyme (peptidyl-dipeptidase A) 1 CAPTOPRIL Protease, Angiotensin Converting Enzyme 93% .13uM NoneNone View
mitogen activated protein kinase 14 TIRILAZAD Protein Serine/Threonine Kinase, p38alpha 93% 7.406uM NoneNone View
mitogen-activated protein kinase 14 TIRILAZAD Protein Serine/Threonine Kinase, p38alpha 93% 7.406uM NoneNone View
Protein-tyrosine kinase, Fyn 2-HYDROXYPROPYL-BETA-CYCLODEXTRIN Protein Tyrosine Kinase, Fyn 93% 3.043uM NoneNone View
calcium channel, voltage-dependent, gamma subunit 8 U-78517F Calcium Channel Type L, Benzothiazepine 93% 1.65uM 1.466uM View
calcium channel, voltage-dependent, gamma subunit 7 U-78517F Calcium Channel Type L, Benzothiazepine 93% 1.65uM 1.466uM View
calcium channel, voltage-dependent, gamma subunit 6 U-78517F Calcium Channel Type L, Benzothiazepine 93% 1.65uM 1.466uM View
calcium channel, voltage-dependent, gamma subunit 5 U-78517F Calcium Channel Type L, Benzothiazepine 93% 1.65uM 1.466uM View
calcium channel, voltage-dependent, gamma subunit 4 U-78517F Calcium Channel Type L, Benzothiazepine 93% 1.65uM 1.466uM View
calcium channel, voltage-dependent, gamma subunit 3 U-78517F Calcium Channel Type L, Benzothiazepine 93% 1.65uM 1.466uM View
calcium channel, voltage-dependent, gamma subunit 2 U-78517F Calcium Channel Type L, Benzothiazepine 93% 1.65uM 1.466uM View
calcium channel, voltage-dependent, gamma subunit 1 U-78517F Calcium Channel Type L, Benzothiazepine 93% 1.65uM 1.466uM View
calcium channel, voltage-dependent, beta 4 subunit U-78517F Calcium Channel Type L, Benzothiazepine 93% 1.65uM 1.466uM View
potassium voltage-gated channel, subfamily H, member 8 THIORIDAZINE Potassium Channel HERG 93% 1.588uM 1.301uM View
potassium voltage-gated channel, subfamily H (eag-related), member 6 THIORIDAZINE Potassium Channel HERG 93% 1.588uM 1.301uM View
potassium voltage-gated channel, subfamily H (eag-related), member 7 THIORIDAZINE Potassium Channel HERG 93% 1.588uM 1.301uM View
potassium voltage-gated channel, subfamily H (eag-related), member 2 THIORIDAZINE Potassium Channel HERG 93% 1.588uM 1.301uM View
potassium voltage-gated channel, subfamily H (eag-related), member 5 THIORIDAZINE Potassium Channel HERG 93% 1.588uM 1.301uM View
potassium voltage-gated channel, subfamily H (eag-related), member 3 THIORIDAZINE Potassium Channel HERG 93% 1.588uM 1.301uM View
potassium voltage-gated channel, subfamily H (eag-related), member 4 THIORIDAZINE Potassium Channel HERG 93% 1.588uM 1.301uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 THIORIDAZINE Potassium Channel HERG 93% 1.588uM 1.301uM View
potassium voltage-gated channel, subfamily H (eag-related), member 1 THIORIDAZINE Potassium Channel HERG 93% 1.588uM 1.301uM View
Cytochrom P450-2D6 monooxygenase BW-723C86 CYP450-2D6 Inhibition 93% 2.7743uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 SULOCTIDIL Serotonin Transporter 93% 1.2532uM .6658uM View
epidermal growth factor receptor SULOCTIDIL Protein Tyrosine Kinase, EGF Receptor 93% .7944uM NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) GLYBURIDE CYP450-2C9 Inhibition 93% 1.602uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 GLYBURIDE CYP450-2C9 Inhibition 93% 1.602uM NoneNone View
androgen receptor HYDROXYPROGESTERONE Testosterone 93% .739uM .493uM View
opioid receptor, sigma 1 TOLPERISONE Sigma1 93% .013uM .005587uM View
5-hydroxytryptamine (serotonin) receptor 2A CINNARIZINE Serotonin 5-HT2A 93% .36uM .103uM View
5-hydroxytryptamine (serotonin) receptor 1A THIORIDAZINE Serotonin 5-HT1A 93% .06uM .034uM View
glycine receptor, alpha 3 DESLORATADINE Glycine, Strychnine-Sensitive 93% .834uM .471uM View
glycine receptor, alpha 1 subunit DESLORATADINE Glycine, Strychnine-Sensitive 93% .834uM .471uM View
glycine receptor, beta subunit DESLORATADINE Glycine, Strychnine-Sensitive 93% .834uM .471uM View
glycine receptor, alpha 2 subunit DESLORATADINE Glycine, Strychnine-Sensitive 93% .834uM .471uM View
dopamine receptor 2 CINNARIZINE Dopamine D2L 93% .776uM .259uM View
Cytochrom P450-2D6 monooxygenase L-744832 CYP450-2D6 Inhibition 93% .7uM NoneNone View
Cytochrome P450, subfamily IIC (mephenytoin 4-hydroxylase) PODOPHYLLOTOXIN CYP450-2C9 Inhibition 93% 4uM NoneNone View
cytochrome P450, family 2, subfamily C, polypeptide 9 PODOPHYLLOTOXIN CYP450-2C9 Inhibition 93% 4uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, dopamine), member 3 BITHIONOL Dopamine Transporter 93% 2.181uM 1.733uM View
cholinergic receptor, muscarinic 2 DIPHENIDOL Muscarinic M2 93% .77uM .274uM View
androgen receptor ETHISTERONE Testosterone 93% .067uM .044uM View
progesterone receptor ETHYLESTRENOL Progesterone 93% .201uM .026uM View
progesterone receptor ETHYLESTRENOL Progesterone 93% .201uM .026uM View
cholinergic receptor, muscarinic 2 ETHYLESTRENOL Muscarinic M2 93% .292uM .104uM View
adrenergic receptor, alpha 1a CLONIDINE Adrenergic alpha1A 93% .372uM .151uM View