Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
potassium voltage-gated channel, subfamily H (eag-related), member 2 HALOPERIDOL Potassium Channel HERG 99% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 5 HALOPERIDOL Potassium Channel HERG 99% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 3 HALOPERIDOL Potassium Channel HERG 99% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 4 HALOPERIDOL Potassium Channel HERG 99% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 1 HALOPERIDOL Potassium Channel HERG 99% NoneNone NoneNone View
potassium voltage-gated channel, subfamily H (eag-related), member 1 HALOPERIDOL Potassium Channel HERG 99% NoneNone NoneNone View
5-hydroxytryptamine (serotonin) receptor 2C BW-723C86 Serotonin 5-HT2C 99% .2043uM .107uM View
opioid receptor, sigma 1 SULOCTIDIL Sigma1 99% .1172uM .0493uM View
calcium channel, voltage-dependent, gamma subunit 8 SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, gamma subunit 7 SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, gamma subunit 6 SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, gamma subunit 5 SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, gamma subunit 4 SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, gamma subunit 3 SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, gamma subunit 2 SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, gamma subunit 1 SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, beta 4 subunit SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, beta 3 subunit SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, beta 2 subunit SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, alpha 1F subunit SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, beta 1 subunit SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 SULOCTIDIL Calcium Channel Type L, Benzothiazepine 99% .1712uM .1522uM View
Cytochrom P450-1A2 monooxygenase HEXACHLOROPHENE CYP450-1A2 Inhibition 99% 1.3133uM NoneNone View
opioid receptor, sigma 1 FLUNARIZINE Sigma1 99% .025uM .01uM View
5-hydroxytryptamine (serotonin) receptor 2C PROPAFENONE Serotonin 5-HT2C 99% .384uM .201uM View
5-hydroxytryptamine (serotonin) receptor 2B DESLORATADINE Serotonin 5-HT2B 99% .043uM .028uM View
5-hydroxytryptamine (serotonin) receptor 2A THIORIDAZINE Serotonin 5-HT2A 99% .004366uM .001247uM View
5-hydroxytryptamine (serotonin) receptor 2A DOMPERIDONE Serotonin 5-HT2A 99% .037uM .011uM View
cholinergic receptor, muscarinic 5 DESLORATADINE Muscarinic M5 99% .292uM .21uM View
cholinergic receptor, muscarinic 3 THIORIDAZINE Muscarinic M3 99% .09uM .019uM View
cholinergic receptor, muscarinic 4 THIORIDAZINE Muscarinic M4 99% .08uM .011uM View
cholinergic receptor, muscarinic 2 THIORIDAZINE Muscarinic M2 99% .106uM .038uM View
cholinergic receptor, muscarinic 2 METHSCOPOLAMINE BROMIDE Muscarinic M2 99% .000422uM .00015uM View
cholinergic receptor, muscarinic 1 METHSCOPOLAMINE BROMIDE Muscarinic M1 99% .001334uM .000321uM View
histamine receptor H 1 FLUNARIZINE Histamine H1, Central 99% .158uM .018uM View
prostaglandin-endoperoxide synthase 1 BROMFENAC Cyclooxygenase COX-1 99% .008481uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) BROMFENAC Cyclooxygenase COX-1 99% .008481uM NoneNone View
Cytochrom P450-2D6 monooxygenase DIPHENIDOL CYP450-2D6 Inhibition 99% .3263uM NoneNone View
ATPase, Na+/K+ transporting, alpha 4 polypeptide PROSCILLARIDIN ATPase, Na+/K+ 99% .088uM NoneNone View
ATPase, Na+/K+ transporting, alpha 3 polypeptide PROSCILLARIDIN ATPase, Na+/K+ 99% .088uM NoneNone View
ATPase, Na+/K+ transporting, alpha 2 polypeptide PROSCILLARIDIN ATPase, Na+/K+ 99% .088uM NoneNone View
ATPase, Na+/K+ transporting, alpha 1 polypeptide PROSCILLARIDIN ATPase, Na+/K+ 99% .088uM NoneNone View
ATPase, Na+/K+ transporting, beta 1 polypeptide PROSCILLARIDIN ATPase, Na+/K+ 99% .088uM NoneNone View
ATPase, Na+/K+ transporting, beta 3 polypeptide PROSCILLARIDIN ATPase, Na+/K+ 99% .088uM NoneNone View
ATPase, Na+/K+ transporting, beta 2 polypeptide PROSCILLARIDIN ATPase, Na+/K+ 99% .088uM NoneNone View
ATPase, (Na+)/K+ transporting, beta 4 polypeptide PROSCILLARIDIN ATPase, Na+/K+ 99% .088uM NoneNone View
cholinergic receptor, muscarinic 5 PIPERILATE ETHOBROMIDE Muscarinic M5 99% .107uM .077uM View
cholinergic receptor, muscarinic 3 PIPERILATE ETHOBROMIDE Muscarinic M3 99% .157uM .033uM View
cholinergic receptor, muscarinic 4 PIPERILATE ETHOBROMIDE Muscarinic M4 99% .062uM .008584uM View
adrenergic receptor, alpha 2a BITHIONOL Adrenergic alpha2A 99% 3.824uM 1.434uM View
adrenergic receptor, alpha 2a ALPHA-ERGOCRYPTINE Adrenergic alpha2A 99% .007946uM .00298uM View
progesterone receptor ETHISTERONE Progesterone 99% .059uM .00775uM View
progesterone receptor ETHISTERONE Progesterone 99% .059uM .00775uM View
5-hydroxytryptamine (serotonin) receptor 1A METHYLERGONOVINE Serotonin 5-HT1A 99% .00407uM .002326uM View
cholinergic receptor, muscarinic 4 BENZTROPINE Muscarinic M4 99% .002385uM .000333uM View
adrenergic receptor, alpha 2b PIPAMAZINE Adrenergic alpha2C 98% .045uM .006468uM View
adrenergic receptor, alpha 2c (Non-specific probe) PIPAMAZINE Adrenergic alpha2C 98% .045uM .006468uM View
calcium channel, voltage-dependent, beta 2 subunit NIMODIPINE Calcium Channel Type L, Dihydropyridine 98% .000242uM .000156uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit NIMODIPINE Calcium Channel Type L, Dihydropyridine 98% .000242uM .000156uM View
calcium channel, voltage-dependent, alpha 1F subunit NIMODIPINE Calcium Channel Type L, Dihydropyridine 98% .000242uM .000156uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit NIMODIPINE Calcium Channel Type L, Dihydropyridine 98% .000242uM .000156uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit NIMODIPINE Calcium Channel Type L, Dihydropyridine 98% .000242uM .000156uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit NIMODIPINE Calcium Channel Type L, Dihydropyridine 98% .000242uM .000156uM View
calcium channel, voltage-dependent, beta 1 subunit NIMODIPINE Calcium Channel Type L, Dihydropyridine 98% .000242uM .000156uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit NIMODIPINE Calcium Channel Type L, Dihydropyridine 98% .000242uM .000156uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit NIMODIPINE Calcium Channel Type L, Dihydropyridine 98% .000242uM .000156uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 NIMODIPINE Calcium Channel Type L, Dihydropyridine 98% .000242uM .000156uM View
acetylcholinesterase (YT blood group) NEOSTIGMINE BROMIDE Acetylcholinesterase 98% .2uM NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase NEOSTIGMINE BROMIDE Acetylcholinesterase 98% .2uM NoneNone View
acetylcholinesterase NEOSTIGMINE BROMIDE Acetylcholinesterase 98% .2uM NoneNone View
adrenergic receptor, alpha 2b OXICONAZOLE Adrenergic alpha2C 98% 4.1645uM .6051uM View
adrenergic receptor, alpha 2c (Non-specific probe) OXICONAZOLE Adrenergic alpha2C 98% 4.1645uM .6051uM View
dopamine receptor D3 OXYBUTYNIN Dopamine D3 98% .4288uM .1456uM View
cholinergic receptor, muscarinic 2 ORPHENADRINE Muscarinic M2 98% .376uM .134uM View
dopamine receptor D3 LEVOSULPIRIDE Dopamine D3 98% .123uM .042uM View
adrenergic receptor, alpha 1a OXYMETAZOLINE Adrenergic alpha1A 98% .038uM .016uM View
adrenergic receptor, alpha 1d (Non-specific probe) PROCHLORPERAZINE Adrenergic alpha1D 98% .034uM .016uM View
calcium channel, voltage-dependent, gamma subunit 8 CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, gamma subunit 7 CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, gamma subunit 6 CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, gamma subunit 5 CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, gamma subunit 4 CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, gamma subunit 3 CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, gamma subunit 2 CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, gamma subunit 1 CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, beta 4 subunit CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, beta 3 subunit CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, beta 2 subunit CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, alpha 1F subunit CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, L type, alpha 1D subunit CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, L type, alpha 1C subunit CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, P/Q type, alpha 1A subunit CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, beta 1 subunit CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, L type, alpha 1E subunit CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 CYPROHEPTADINE Calcium Channel Type L, Benzothiazepine 98% 1.925uM 1.711uM View
carbonic anhydrase 5a, mitochondrial PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase 3 PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase 2 PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase 4 PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase XI PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase IX PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase VIII PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase VII PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase VA, mitochondrial PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase IV PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase III, muscle specific PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase I PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase XIV PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase VB, mitochondrial PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase XII PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase VI PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
carbonic anhydrase II PIOGLITAZONE Carbonic Anhydrase 98% .114uM NoneNone View
nuclear receptor subfamily 3, group C, member 1 FLUOROMETHOLONE Glucocorticoid 98% .003471uM .001578uM View
5-hydroxytryptamine (serotonin) receptor 2C CYPROHEPTADINE Serotonin 5-HT2C 98% .00244uM .001278uM View
dopamine receptor D1A CYPROHEPTADINE Dopamine D1 98% .158uM .079uM View
cholinergic receptor, muscarinic 5 CYPROHEPTADINE Muscarinic M5 98% .003835uM .002755uM View
dopamine receptor 2 METOCLOPRAMIDE Dopamine D2L 98% .127uM .042uM View
cholinergic receptor, muscarinic 3 HOMATROPINE HYDROBROMIDE Muscarinic M3 98% .076uM .016uM View
cholinergic receptor, muscarinic 5 HOMATROPINE HYDROBROMIDE Muscarinic M5 98% .055uM .039uM View
dopamine receptor 2 PIPAMAZINE Dopamine D2L 98% .00405uM .00135uM View
adenosine A1 receptor ECONAZOLE Adenosine A1 98% 16.924uM 9.872uM View
cholinergic receptor, muscarinic 3 MICONAZOLE Muscarinic M3 98% 3.154uM .668uM View
adenosine A1 receptor MICONAZOLE Adenosine A1 98% 12.519uM 7.303uM View
mu-opioid receptor MOR MICONAZOLE Opiate mu 98% 6.059uM 2.46uM View
cholinergic receptor, muscarinic 1 DEXCHLORPHENIRAMINE Muscarinic M1 98% 1.383uM .333uM View
adrenergic receptor, alpha 2a ERGOCORNINE Adrenergic alpha2A 98% .006296uM .002361uM View
3-hydroxy-3-methylglutaryl-Coenzyme A reductase MEVASTATIN HMG-CoA Reductase 98% .119uM NoneNone View
Cytochrom P450-2C19 monooxygenase HEXACHLOROPHENE CYP450-2C19 Inhibition 98% 1.2265uM NoneNone View
acetylcholinesterase (YT blood group) HEXACHLOROPHENE Acetylcholinesterase 98% 3.0149uM NoneNone View
sodium channel, nonvoltage-gated 1 alpha CLOTRIMAZOLE Sodium Channel, Site 2 98% 6.771uM 6.071uM View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase HEXACHLOROPHENE Acetylcholinesterase 98% 3.0149uM NoneNone View
acetylcholinesterase HEXACHLOROPHENE Acetylcholinesterase 98% 3.0149uM NoneNone View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 METHAPYRILENE Serotonin Transporter 98% .2uM .106uM View
5-hydroxytryptamine (serotonin) receptor 2C METHAPYRILENE Serotonin 5-HT2C 98% .744uM .39uM View
5-hydroxytryptamine (serotonin) receptor 2A TERFENADINE Serotonin 5-HT2A 98% .255uM .073uM View
5-hydroxytryptamine (serotonin) receptor 2A CYCLIZINE Serotonin 5-HT2A 98% .225uM .064uM View
lymphocyte protein tyrosine kinase (mapped) IODOQUINOL Protein Tyrosine Kinase, Lck 98% 2.461uM NoneNone View
cholinergic receptor, muscarinic 5 THIORIDAZINE Muscarinic M5 98% .009246uM .006643uM View
cholinergic receptor, muscarinic 5 VALETHAMATE BROMIDE Muscarinic M5 98% .034uM .024uM View
cholinergic receptor, muscarinic 2 DESLORATADINE Muscarinic M2 98% .107uM .038uM View
cholinergic receptor, muscarinic 1 DIMENHYDRINATE Muscarinic M1 98% .451uM .109uM View
cysteinyl leukotriene receptor 1 ZAFIRLUKAST Leukotriene D4 98% .001731uM .000865uM View
cysteinyl leukotriene receptor 1 ZAFIRLUKAST Leukotriene D4 98% .001731uM .000865uM View
histamine receptor H 1 THIORIDAZINE Histamine H1, Central 98% .072uM .008412uM View
histamine receptor H 1 CINNARIZINE Histamine H1, Central 98% .074uM .008622uM View
dopamine receptor 2 DOMPERIDONE Dopamine D2L 98% .002647uM .000882uM View
dopamine receptor D1A THIORIDAZINE Dopamine D1 98% .194uM .097uM View
Cytochrom P450-2D6 monooxygenase BOPINDOLOL CYP450-2D6 Inhibition 98% 5.4764uM NoneNone View
Cytochrom P450-2D6 monooxygenase PERGOLIDE CYP450-2D6 Inhibition 98% .2uM NoneNone View
Cytochrom P450-2C19 monooxygenase IDEBENONE CYP450-2C19 Inhibition 98% .8uM NoneNone View
mitogen activated protein kinase 14 BITHIONOL Protein Serine/Threonine Kinase, p38alpha 98% .318uM NoneNone View
mitogen-activated protein kinase 14 BITHIONOL Protein Serine/Threonine Kinase, p38alpha 98% .318uM NoneNone View
adrenergic receptor, alpha 2b BERBERINE CHLORIDE Adrenergic alpha2B 98% .601uM .274uM View
cholinergic receptor, muscarinic 4 DIPHENIDOL Muscarinic M4 98% .271uM .038uM View
androgen receptor MEDROXYPROGESTERONE ACETATE Testosterone 98% .007259uM .004839uM View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) BITHIONOL Protein Tyrosine Kinase, HER2 Receptor 98% 2.147uM NoneNone View
A3 adenosine receptor BITHIONOL Adenosine A3 98% .829uM .468uM View
v-erb-b2 erythroblastic leukemia viral oncogene homolog 2, neuro/glioblastoma derived oncogene homolog (avian) BITHIONOL Protein Tyrosine Kinase, HER2 Receptor 98% 2.147uM NoneNone View
nuclear receptor subfamily 3, group C, member 1 MEDROXYPROGESTERONE ACETATE Glucocorticoid 98% .019uM .008637uM View
5-hydroxytryptamine (serotonin) receptor 2C ALPHA-ERGOCRYPTINE Serotonin 5-HT2C 98% .147uM .077uM View
dopamine receptor D3 METHYLERGONOVINE Dopamine D3 98% .167uM .057uM View
5-hydroxytryptamine (serotonin) receptor 2C METHYLERGONOVINE Serotonin 5-HT2C 98% .013uM .006558uM View
5-hydroxytryptamine (serotonin) receptor 2A METHYLERGONOVINE Serotonin 5-HT2A 98% .002547uM .000728uM View
adrenergic receptor, alpha 1a DOBUTAMINE Adrenergic alpha1A 98% .11uM .045uM View
cholinergic receptor, muscarinic 5 MAPROTILINE Muscarinic M5 98% .16uM .115uM View
adrenergic receptor, beta 1 (S)-(-)-PINDOLOL Adrenergic beta1 98% .000752uM .000434uM View
adrenergic, beta-1-, receptor (S)-(-)-PINDOLOL Adrenergic beta1 98% .000752uM .000434uM View
adrenergic receptor, alpha 1b LISURIDE Adrenergic alpha1B 98% .121uM .067uM View
dopamine receptor 2 ERGOTAMINE Dopamine D2L 98% .0043uM .001433uM View
adrenergic receptor, alpha 1a DOMPERIDONE Adrenergic alpha1A 98% .285uM .116uM View
5-hydroxytryptamine (serotonin) receptor 1A ERGOTAMINE Serotonin 5-HT1A 98% .000774uM .000443uM View
adrenergic receptor, alpha 2b ERGOTAMINE Adrenergic alpha2C 98% .012uM .001809uM View
adrenergic receptor, alpha 2c (Non-specific probe) ERGOTAMINE Adrenergic alpha2C 98% .012uM .001809uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 PYRILAMINE Serotonin Transporter 98% .047uM .025uM View
adrenergic receptor, alpha 2a PROMAZINE Adrenergic alpha2A 98% .337uM .126uM View
cholinergic receptor, muscarinic 5 PROMAZINE Muscarinic M5 98% .064uM .046uM View
sodium channel, voltage-gated, type X, alpha CLOTRIMAZOLE Sodium Channel, Site 2 98% 6.771uM 6.071uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 PROMAZINE Serotonin Transporter 98% .086uM .046uM View
adrenergic receptor, alpha 2b PROMAZINE Adrenergic alpha2C 98% .253uM .037uM View
adrenergic receptor, alpha 2c (Non-specific probe) PROMAZINE Adrenergic alpha2C 98% .253uM .037uM View
cholinergic receptor, muscarinic 4 PROMAZINE Muscarinic M4 98% .299uM .042uM View
cholinergic receptor, muscarinic 4 PAROXETINE Muscarinic M4 98% .244uM .034uM View
gamma-aminobutyric acid A receptor, alpha 1 ZOPICLONE GABAA, Benzodiazepine, Central 98% .125uM .102uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 2 ZOPICLONE GABAA, Benzodiazepine, Central 98% .125uM .102uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 1 ZOPICLONE GABAA, Benzodiazepine, Central 98% .125uM .102uM View
gamma-aminobutyric acid A receptor, delta ZOPICLONE GABAA, Benzodiazepine, Central 98% .125uM .102uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 3 ZOPICLONE GABAA, Benzodiazepine, Central 98% .125uM .102uM View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase OXICONAZOLE Acetylcholinesterase 97% 4.6465uM NoneNone View
acetylcholinesterase OXICONAZOLE Acetylcholinesterase 97% 4.6465uM NoneNone View
Protein-tyrosine kinase, Fyn EBASTINE Protein Tyrosine Kinase, Fyn 97% .8101uM NoneNone View
adrenergic receptor, alpha 2b EBASTINE Adrenergic alpha2B 97% .7389uM .3373uM View
5-hydroxytryptamine (serotonin) receptor 2B EBASTINE Serotonin 5-HT2B 97% .3126uM .1989uM View