Gene Activity List


Gene Activity List

Gene Compound Assay Inh Ic50 Ki View
adrenergic receptor, alpha 2a MIANSERIN Adrenergic alpha2A 99% .043uM .016uM View
5-hydroxytryptamine (serotonin) receptor 2A MIANSERIN Serotonin 5-HT2A 99% .001764uM .000504uM View
5-hydroxytryptamine (serotonin) receptor 1B LYSERGOL Serotonin 5-HT1B 99% .002977uM .001353uM View
5-hydroxytryptamine (serotonin) receptor 2A METHYSERGIDE Serotonin 5-HT2A 99% .013uM .003832uM View
5-hydroxytryptamine (serotonin) receptor 2C LYSERGOL Serotonin 5-HT2C 99% .034uM .018uM View
cholinergic receptor, muscarinic 1 MEPAZINE Muscarinic M1 99% .079uM .019uM View
adrenergic receptor, alpha 1a MEPAZINE Adrenergic alpha1A 99% .144uM .058uM View
mitogen activated protein kinase 14 RWJ-68354 Protein Serine/Threonine Kinase, p38alpha 99% .075uM NoneNone View
mitogen-activated protein kinase 14 RWJ-68354 Protein Serine/Threonine Kinase, p38alpha 99% .075uM NoneNone View
monoamine oxidase A 2-ACETYLAMINOFLUORENE Monoamine Oxidase MAOA 99% .059uM NoneNone View
monoamine oxidase A 2-ACETYLAMINOFLUORENE Monoamine Oxidase MAOA 99% .059uM NoneNone View
Protein-tyrosine kinase, Fyn LEAD (II) ACETATE Protein Tyrosine Kinase, Fyn 99% .431uM NoneNone View
adrenergic receptor, beta 1 PROPRANOLOL Adrenergic beta1 99% .002543uM .001468uM View
adrenergic, beta-1-, receptor PROPRANOLOL Adrenergic beta1 99% .002543uM .001468uM View
prostaglandin-endoperoxide synthase 1 N,N'-DIPHENYL-P-PHENYLENEDIAMINE Cyclooxygenase COX-1 99% .26uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) N,N'-DIPHENYL-P-PHENYLENEDIAMINE Cyclooxygenase COX-1 99% .26uM NoneNone View
cholinergic receptor, muscarinic 4 MITOXANTRONE Muscarinic M4 99% .6441uM .0898uM View
5-hydroxytryptamine (serotonin) receptor 2B RISPERIDONE Serotonin 5-HT2B 99% .023uM .015uM View
dopamine receptor D3 QUINACRINE Dopamine D3 99% 1.318uM .448uM View
prostaglandin-endoperoxide synthase 1 DEXKETOPROFEN Cyclooxygenase COX-1 99% .004483uM NoneNone View
prostaglandin-endoperoxide synthase 1 (prostaglandin G/H synthase and cyclooxygenase) DEXKETOPROFEN Cyclooxygenase COX-1 99% .004483uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 2A KETOTIFEN Serotonin 5-HT2A 99% .031uM .008977uM View
acetylcholinesterase (YT blood group) PHYSOSTIGMINE Acetylcholinesterase 99% .175uM NoneNone View
collagen-like tail subunit (single strand of homotrimer) of asymmetric acetylcholinesterase PHYSOSTIGMINE Acetylcholinesterase 99% .175uM NoneNone View
acetylcholinesterase PHYSOSTIGMINE Acetylcholinesterase 99% .175uM NoneNone View
adrenergic receptor, beta 2 BOPINDOLOL Adrenergic beta2 99% .02uM .014uM View
5-hydroxytryptamine (serotonin) receptor 1A BOPINDOLOL Serotonin 5-HT1A 99% .267uM .153uM View
cholinergic receptor, muscarinic 4 NORTRIPTYLINE Muscarinic M4 99% .095uM .013uM View
protein kinase C, delta FAMOTIDINE Phorbol Ester 3% NoneNone NoneNone View
sodium channel, voltage-gated, type IV, beta RITONAVIR Sodium Channel, Site 2 99% 2.379uM 2.133uM View
sodium channel associated protein 1 RITONAVIR Sodium Channel, Site 2 99% 2.379uM 2.133uM View
sodium channel associated protein 2 RITONAVIR Sodium Channel, Site 2 99% 2.379uM 2.133uM View
sodium channel, voltage-gated, type III, beta RITONAVIR Sodium Channel, Site 2 99% 2.379uM 2.133uM View
sodium channel, voltage-gated, type I, alpha RITONAVIR Sodium Channel, Site 2 99% 2.379uM 2.133uM View
sodium channel, voltage-gated, type IX, alpha RITONAVIR Sodium Channel, Site 2 99% 2.379uM 2.133uM View
sodium channel, voltage-gated, type VII, alpha RITONAVIR Sodium Channel, Site 2 99% 2.379uM 2.133uM View
amiloride-sensitive cation channel 5, intestinal RITONAVIR Sodium Channel, Site 2 99% 2.379uM 2.133uM View
sodium channel, voltage-gated, type III, beta RITONAVIR Sodium Channel, Site 2 99% 2.379uM 2.133uM View
calcium channel, voltage-dependent, beta 3 subunit AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, beta 2 subunit AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, L type, alpha 1S subunit AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, alpha 1F subunit AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
5-hydroxytryptamine receptor 6 CHLORPROMAZINE Serotonin 5-HT6 99% .057uM .026uM View
Protein-tyrosine kinase, Fyn GOLD SODIUM THIOMALATE Protein Tyrosine Kinase, Fyn 99% .811uM NoneNone View
cholinergic receptor, muscarinic 3 TROPICAMIDE Muscarinic M3 99% .142uM .03uM View
cholinergic receptor, muscarinic 5 TROPICAMIDE Muscarinic M5 99% .089uM .064uM View
arachidonate 15-lipoxygenase, second type CATECHOL Lipoxygenase 15-LO 99% .868uM NoneNone View
arachidonate 15-lipoxygenase CATECHOL Lipoxygenase 15-LO 99% .868uM NoneNone View
arachidonate 15-lipoxygenase CATECHOL Lipoxygenase 15-LO 99% .868uM NoneNone View
adrenergic receptor, alpha 1a DIHYDROERGOTAMINE Adrenergic alpha1A 99% .005028uM .002035uM View
5-hydroxytryptamine (serotonin) receptor 1A DIHYDROERGOTAMINE Serotonin 5-HT1A 99% .000659uM .000377uM View
5-hydroxytryptamine (serotonin) receptor 2A DIHYDROERGOTAMINE Serotonin 5-HT2A 99% .007955uM .002273uM View
5-hydroxytryptamine (serotonin) receptor 2B YOHIMBINE Serotonin 5-HT2B 99% .074uM .047uM View
cholinergic receptor, muscarinic 5 TAMOXIFEN Muscarinic M5 99% 2.585uM 1.857uM View
cholinergic receptor, muscarinic 1 TAMOXIFEN Muscarinic M1 99% 2.829uM .681uM View
cholinergic receptor, muscarinic 4 TAMOXIFEN Muscarinic M4 99% 4.817uM .672uM View
dopamine receptor D1A TAMOXIFEN Dopamine D1 99% 8.502uM 4.251uM View
5-hydroxytryptamine (serotonin) receptor 2C DIHYDROERGOTAMINE Serotonin 5-HT2C 99% .09uM .047uM View
cholinergic receptor, muscarinic 1 DICYCLOMINE Muscarinic M1 99% .003463uM .000834uM View
5-hydroxytryptamine (serotonin) receptor 2A ERGONOVINE Serotonin 5-HT2A 99% .002205uM .00063uM View
5-hydroxytryptamine (serotonin) receptor 2A CISAPRIDE Serotonin 5-HT2A 99% .003856uM .001102uM View
cholinergic receptor, muscarinic 2 DICYCLOMINE Muscarinic M2 99% .046uM .016uM View
adrenergic receptor, alpha 1b CLOMIPRAMINE Adrenergic alpha1B 99% .132uM .073uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 CLOMIPRAMINE Adrenergic, Norepinephrine Transporter 99% .071uM .07uM View
5-hydroxytryptamine receptor 6 CLOMIPRAMINE Serotonin 5-HT6 99% .245uM .114uM View
cholinergic receptor, muscarinic 2 ATROPINE Muscarinic M2 99% .003735uM .001328uM View
cholinergic receptor, muscarinic 3 CLOMIPRAMINE Muscarinic M3 99% .17uM .036uM View
cholinergic receptor, muscarinic 4 CLOMIPRAMINE Muscarinic M4 99% .091uM .013uM View
5-hydroxytryptamine (serotonin) receptor 2C CLOZAPINE Serotonin 5-HT2C 99% .006039uM .003163uM View
adrenergic receptor, alpha 2b CLOZAPINE Adrenergic alpha2C 99% .007875uM .001144uM View
adrenergic receptor, alpha 2c (Non-specific probe) CLOZAPINE Adrenergic alpha2C 99% .007875uM .001144uM View
5-hydroxytryptamine (serotonin) receptor 1A CARVEDILOL Serotonin 5-HT1A 99% .005842uM .003338uM View
cholinergic receptor, muscarinic 3 CLOZAPINE Muscarinic M3 99% .078uM .017uM View
cholinergic receptor, muscarinic 4 CLOZAPINE Muscarinic M4 99% .045uM .006303uM View
5-hydroxytryptamine receptor 6 CLOZAPINE Serotonin 5-HT6 99% .011uM .005055uM View
dopamine receptor 2 CARVEDILOL Dopamine D2L 99% .146uM .049uM View
cholinergic receptor, muscarinic 3 CLEMASTINE Muscarinic M3 99% .039uM .008253uM View
cholinergic receptor, muscarinic 4 CLEMASTINE Muscarinic M4 99% .02uM .002773uM View
adrenergic receptor, alpha 2a CARVEDILOL Adrenergic alpha2A 99% .106uM .04uM View
adrenergic receptor, beta 3 CARVEDILOL Adrenergic beta3 99% .004155uM .003116uM View
dopamine receptor D3 CARVEDILOL Dopamine D3 99% .577uM .196uM View
histamine receptor H 1 CLOZAPINE Histamine H1, Central 99% .004912uM .000571uM View
5-hydroxytryptamine (serotonin) receptor 2B CLOMIPRAMINE Serotonin 5-HT2B 99% .239uM .152uM View
5-hydroxytryptamine (serotonin) receptor 2A CARVEDILOL Serotonin 5-HT2A 99% .41uM .117uM View
nuclear receptor subfamily 3, group C, member 1 CHLORMADINONE ACETATE Glucocorticoid 99% .0377uM .0172uM View
solute carrier family 28 (sodium-coupled nucleoside transporter), member 3 DIPYRIDAMOLE Adenosine Transporter 99% .083uM .029uM View
concentrative Na+ nucleoside cotransporter (DBSS) DIPYRIDAMOLE Adenosine Transporter 99% .083uM .029uM View
solute carrier family 28 (sodium-coupled nucleoside transporter), member 1 DIPYRIDAMOLE Adenosine Transporter 99% .083uM .029uM View
adenine nucleotide translocase (DBSS) (Non-specific probe) DIPYRIDAMOLE Adenosine Transporter 99% .083uM .029uM View
solute carrier family 25 (mitochondrial carrier; adenine nucleotide translocator), member 4 DIPYRIDAMOLE Adenosine Transporter 99% .083uM .029uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 4 FLUMAZENIL GABAA, Benzodiazepine, Central 99% .003867uM .003151uM View
gamma-aminobutyric acid A receptor, gamma 1 FLUMAZENIL GABAA, Benzodiazepine, Central 99% .003867uM .003151uM View
gamma-aminobutyric acid A receptor, pi FLUMAZENIL GABAA, Benzodiazepine, Central 99% .003867uM .003151uM View
AT hook, DNA binding motif, containing 1 (DBSS) FLUMAZENIL GABAA, Benzodiazepine, Central 99% .003867uM .003151uM View
gamma-aminobutyric acid A receptor, theta FLUMAZENIL GABAA, Benzodiazepine, Central 99% .003867uM .003151uM View
gamma-aminobutyric acid A receptor, gamma 2 FLUMAZENIL GABAA, Benzodiazepine, Central 99% .003867uM .003151uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 6 FLUMAZENIL GABAA, Benzodiazepine, Central 99% .003867uM .003151uM View
calcium channel, voltage-dependent, N type, alpha 1B subunit AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, alpha2/delta subunit 1 AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, gamma subunit 8 AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, gamma subunit 7 AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, gamma subunit 6 AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, gamma subunit 5 AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, gamma subunit 4 AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, gamma subunit 3 AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, gamma subunit 2 AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, gamma subunit 1 AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
calcium channel, voltage-dependent, beta 4 subunit AMIODARONE Calcium Channel Type L, Dihydropyridine 99% .165uM .106uM View
adrenergic receptor, alpha 1a BENZTROPINE Adrenergic alpha1A 99% .142uM .057uM View
cholinergic receptor, muscarinic 5 BENZTROPINE Muscarinic M5 99% .002019uM .001451uM View
5-hydroxytryptamine (serotonin) receptor 2A BENZTROPINE Serotonin 5-HT2A 99% .024uM .006968uM View
5-hydroxytryptamine (serotonin) receptor 2C MAPROTILINE Serotonin 5-HT2C 99% .078uM .041uM View
adrenergic receptor, alpha 2b MAPROTILINE Adrenergic alpha2B 99% .292uM .133uM View
angiotensin 1 converting enzyme 1 LISINOPRIL Protease, Angiotensin Converting Enzyme 99% .006038uM NoneNone View
angiotensin I converting enzyme (peptidyl-dipeptidase A) 1 LISINOPRIL Protease, Angiotensin Converting Enzyme 99% .006038uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 1A LISURIDE Serotonin 5-HT1A 99% .000465uM .000266uM View
5-hydroxytryptamine (serotonin) receptor 1B LISURIDE Serotonin 5-HT1B 99% .01uM .004594uM View
5-hydroxytryptamine (serotonin) receptor 2A DIHYDROERGOCRISTINE MESYLATE Serotonin 5-HT2A 99% .015uM .00424uM View
adrenergic receptor, alpha 1d (Non-specific probe) ERGOTAMINE Adrenergic alpha1D 99% .049uM .024uM View
adrenergic receptor, alpha 1a DIHYDROERGOCRISTINE MESYLATE Adrenergic alpha1A 99% .00162uM .000656uM View
adrenergic receptor, alpha 1a QUETIAPINE Adrenergic alpha1A 99% .0862uM .0349uM View
cholinergic receptor, muscarinic 1 PROMAZINE Muscarinic M1 99% .487uM .117uM View
cholinergic receptor, muscarinic 3 PAROXETINE Muscarinic M3 99% .179uM .038uM View
androgen receptor 17-METHYLTESTOSTERONE Testosterone 99% .006399uM .004266uM View
5-hydroxytryptamine (serotonin) receptor 2A METERGOLINE Serotonin 5-HT2A 99% .000395uM .000113uM View
adrenergic receptor, alpha 1b METERGOLINE Adrenergic alpha1B 99% .262uM .145uM View
adrenergic receptor, alpha 1b THIORIDAZINE Adrenergic alpha1B 99% .004692uM .002597uM View
5-hydroxytryptamine (serotonin) receptor 2A PERGOLIDE Serotonin 5-HT2A 99% .014uM .003904uM View
adrenergic receptor, alpha 1a PROCHLORPERAZINE Adrenergic alpha1A 99% .032uM .013uM View
adrenergic receptor, beta 1 PINDOLOL Adrenergic beta1 99% .000921uM .000532uM View
adrenergic, beta-1-, receptor PINDOLOL Adrenergic beta1 99% .000921uM .000532uM View
5-hydroxytryptamine (serotonin) receptor 2C GUANABENZ Serotonin 5-HT2C 99% .204uM .107uM View
cholinergic receptor, muscarinic 3 CYPROHEPTADINE Muscarinic M3 99% .046uM .009655uM View
progesterone receptor HALCINONIDE Progesterone 99% .00093uM .000121uM View
progesterone receptor HALCINONIDE Progesterone 99% .00093uM .000121uM View
adrenergic receptor, alpha 2a GUANABENZ Adrenergic alpha2A 99% .041uM .015uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 4 LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
gamma-aminobutyric acid A receptor, gamma 1 LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
gamma-aminobutyric acid A receptor, pi LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
AT hook, DNA binding motif, containing 1 (DBSS) LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
gamma-aminobutyric acid A receptor, theta LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
gamma-aminobutyric acid A receptor, gamma 2 LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 6 LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 5 LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
gamma-aminobutyric acid A receptor, alpha 2 LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
gamma-aminobutyric acid A receptor, alpha 1 LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 2 LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 1 LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
gamma-aminobutyric acid A receptor, delta LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 3 LORAZEPAM GABAA, Benzodiazepine, Central 99% .006354uM .005177uM View
cholinergic receptor, muscarinic 2 CYPROHEPTADINE Muscarinic M2 99% .035uM .012uM View
gamma-aminobutyric acid (GABA-A) receptor, subunit alpha 5 FLUMAZENIL GABAA, Benzodiazepine, Central 99% .003867uM .003151uM View
gamma-aminobutyric acid A receptor, alpha 2 FLUMAZENIL GABAA, Benzodiazepine, Central 99% .003867uM .003151uM View
gamma-aminobutyric acid A receptor, alpha 1 FLUMAZENIL GABAA, Benzodiazepine, Central 99% .003867uM .003151uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 2 FLUMAZENIL GABAA, Benzodiazepine, Central 99% .003867uM .003151uM View
gamma-aminobutyric acid (GABA-C) receptor, subunit rho 1 FLUMAZENIL GABAA, Benzodiazepine, Central 99% .003867uM .003151uM View
estrogen receptor 1 ETHINYLESTRADIOL Estrogen ERalpha 99% .000448uM .000128uM View
estrogen receptor 1 ETHINYLESTRADIOL Estrogen ERalpha 99% .000448uM .000128uM View
estrogen receptor 1 ESTRONE Estrogen ERalpha 99% .007647uM .002185uM View
estrogen receptor 1 ESTRONE Estrogen ERalpha 99% .007647uM .002185uM View
adrenergic receptor, alpha 2a 4-OCTYLPHENOL Adrenergic alpha2A 99% 14.288uM 5.358uM View
lymphocyte protein tyrosine kinase (mapped) LIPOPOLYSACCHARIDE E. COLI O55:B5 Protein Tyrosine Kinase, Lck 99% .2938uM NoneNone View
cholinergic receptor, muscarinic 3 4-OCTYLPHENOL Muscarinic M3 99% 19.004uM 4.028uM View
cholinergic receptor, muscarinic 2 4-OCTYLPHENOL Muscarinic M2 99% 12.466uM 4.432uM View
nuclear receptor subfamily 3, group C, member 1 PROGESTERONE Glucocorticoid 99% .33uM .15uM View
arachidonate 15-lipoxygenase, second type BISPHENOL A Lipoxygenase 15-LO 99% 1.304uM NoneNone View
arachidonate 15-lipoxygenase BISPHENOL A Lipoxygenase 15-LO 99% 1.304uM NoneNone View
arachidonate 15-lipoxygenase BISPHENOL A Lipoxygenase 15-LO 99% 1.304uM NoneNone View
carbonic anhydrase 5a, mitochondrial CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase 3 CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase 2 CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase 4 CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase XI CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase IX CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase VIII CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase VII CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase VA, mitochondrial CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase IV CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase III, muscle specific CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase I CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase XIV CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase VB, mitochondrial CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase XII CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase VI CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
carbonic anhydrase II CELECOXIB Carbonic Anhydrase 99% .181uM NoneNone View
Protein-tyrosine kinase, Fyn TIRILAZAD Protein Tyrosine Kinase, Fyn 99% 1.116uM NoneNone View
Cytochrom P450-1A2 monooxygenase ALPHA-NAPHTHOFLAVONE CYP450-1A2 Inhibition 99% .9909uM NoneNone View
adrenergic receptor, alpha 2b AMITRIPTYLINE Adrenergic alpha2C 99% .059uM .008599uM View
adrenergic receptor, alpha 2c (Non-specific probe) AMITRIPTYLINE Adrenergic alpha2C 99% .059uM .008599uM View
cholinergic receptor, muscarinic 1 AMITRIPTYLINE Muscarinic M1 99% .011uM .002724uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 AMITRIPTYLINE Serotonin Transporter 99% .001661uM .000882uM View
solute carrier family 6 (neurotransmitter transporter, serotonin), member 4 AMOXAPINE Serotonin Transporter 99% .034uM .018uM View
adrenergic receptor, alpha 1a AMITRIPTYLINE Adrenergic alpha1A 99% .014uM .005599uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 AMITRIPTYLINE Adrenergic, Norepinephrine Transporter 99% .023uM .022uM View
adrenergic receptor, alpha 1a AMOXAPINE Adrenergic alpha1A 99% .357uM .144uM View
solute carrier family 6 (neurotransmitter transporter, noradrenalin), member 2 AMOXAPINE Adrenergic, Norepinephrine Transporter 99% .013uM .013uM View
5-hydroxytryptamine receptor 6 CLOTRIMAZOLE Serotonin 5-HT6 99% 12.543uM 5.824uM View
cytochrome P450, family 3, subfamily a, polypeptide 13 CLOTRIMAZOLE CYP450-3A4 Inhibition 99% .016uM NoneNone View
5-hydroxytryptamine (serotonin) receptor 2A CHLORPROMAZINE Serotonin 5-HT2A 99% .003851uM .0011uM View
dopamine receptor 2 CHLORPROMAZINE Dopamine D2L 99% .054uM .018uM View